Drugs / JNJ-54175446
last change Jun 2024 re-read 2 minutes ago

JNJ-54175446

Small molecule targets P2RX7 via inhibition

Developed for
major depressive disorder
Investigated by
Janssen Research & Development, LLC · Janssen-Cilag International NV

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT03088644 Mar → Nov 2017 Janssen-Cilag International NV Completed No outcome recorded
Phase 1 NCT03058419 Mar → May 2017 Janssen Research & Development, LLC Completed No outcome recorded
Phase 1 NCT02902601 Oct 2016 → Jun 2017 major depressive disorder Janssen Research & Development, LLC Completed No outcome recorded
Phase 1 NCT02930694 Oct → Dec 2016 Janssen Research & Development, LLC Completed No outcome recorded
Phase 1 NCT02933762 Sep → Nov 2016 Janssen Research & Development, LLC Completed No outcome recorded
Phase 1 NCT02515955 Aug 2015 → Mar 2016 Janssen-Cilag International NV Completed No outcome recorded
Phase 1 NCT02475148 Jun → Oct 2015 Janssen-Cilag International NV Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT04116606 Comparator Sep 2019 → Dec 2023 major depressive disorder CCTU-Core Unknown No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as JNJ-54175446 “A Study to Investigate Safety and Tolerability, Pharmacokinetics, Pharmacodynamics and Food Effect of JNJ-54175446 in Healthy Participants” NCT02475148
7

NCT03058419

NCT02930694

NCT02933762

NCT04116606

NCT02515955

NCT02902601

NCT03088644

Action Inhibit “antagonist of the adenosine triphosphate (ATP)-gated P2X7 channel” NCT04116606
1

“P2X purinoceptor 7 antagonist” CHEMBL4079239

Modality Small molecule CHEMBL4079239
Route Oral “after single oral dose administration” NCT02475148
Target P2RX7 “P2X purinoceptor 7 antagonist” CHEMBL4079239