Drugs / Diquafosol tetrasodium
last change Nov 2023 re-read 2 minutes ago

Diquafosol tetrasodium

also known as DE-089 · Diquafosol · DQS · INS365

Oligonucleotide (other) targets P2RY2 via activation

Developed for
dry eye syndrome
Investigated by
He Eye Hospital · Santen Pharmaceutical Co., Ltd. · Merck Sharp & Dohme LLC

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT03216096 Sep 2017 → Feb 2018 dry eye syndrome Santen Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 21 trial
Phase 2 NCT01189032 ? → Jul 2006 dry eye syndrome Santen Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 33 trials
Phase 3 NCT00037661 Apr 2002 → Mar 2003 dry eye syndrome Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 3 NCT00404131 Mar → Dec 2001 dry eye syndrome Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 3 NCT01240382 ? → Feb 2008 dry eye syndrome Santen Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase not applicable4 trials
NCT05720754 Apr → Jul 2023 dry eye syndrome He Eye Hospital Unknown No outcome recorded
NCT04980144 Mar → Aug 2023 He Eye Hospital Unknown No outcome recorded
NCT05694026 Mar → Jul 2023 dry eye syndrome He Eye Hospital Completed No outcome recorded
NCT05682547 Dec 2022 → Jun 2023 He Eye Hospital Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
NCT02618304 Background Apr 2015 → Feb 2016 eye adnexa disorder Yonsei University Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as Diquafosol tetrasodium “3% Diquafosol Tetrasodium eye drops” NCT02618304
5

NCT05720754

NCT04980144

NCT05694026

NCT00404131

NCT05682547

Known as DE-089 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01240382
2

NCT01189032

NCT03216096

Known as Diquafosol Diquafosol is a P2Y2 receptor agonist that has been shown to be effective in the treatment of dry eye disease (DED)” PMID 31834617 Dec 2019
1

Diquafosol ophthalmic solution (DQS) stimulates P2Y2 receptors on the ocular surface” NCT04980144

Known as DQS “Diquafosol ophthalmic solution (DQS) stimulates P2Y2 receptors on the ocular surface” NCT04980144
1

“Diquafosol ophthalmic solution (DQS) stimulates P2Y2 receptors on the ocular surface” NCT05682547

Known as INS365 “Double-masked, placebo-controlled safety and efficacy trial of diquafosol tetrasodium (INS365) ophthalmic solution for the treatment of dry eye.” PMID 15502479 Nov 2004
1

NCT00037661

Action Activate “a P2Y2 receptor agonist that stimulates fluid and mucin secretion on the ocular surface” PMID 15502479 Nov 2004
Modality Oligonucleotide (other) “Diquafosol tetrasodium is a dinucleotide polyphosphate” NCT04980144
Route Topical “when applied topically in subjects with dry eye disease” NCT00404131
Target P2RY2 “Diquafosol ophthalmic solution (DQS) stimulates P2Y2 receptors on the ocular surface” NCT04980144