Drugs / Epelsiban
last change Oct 2016 re-read 2 minutes ago

Epelsiban

Small molecule targets OXTR via inhibition

Developed for
adenomyosis · premature ejaculation
Investigated by
GlaxoSmithKline

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT02703181 Jul → Sep 2015 GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT02257359 Dec 2014 → Jan 2015 GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT02213029 Aug 2014 → Feb 2016 GlaxoSmithKline Terminated No outcome recorded
Phase 1 NCT01669083 Aug 2012 → Mar 2013 GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT00549211 Oct 2007 → ? pregnancy disorder, premature ejaculation GlaxoSmithKline Completed No outcome recorded
Phase 21 trial
Phase 2 NCT02794467 Jul → Oct 2016 adenomyosis GlaxoSmithKline Withdrawn No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01021553 Comparator Dec 2009 → May 2011 premature ejaculation GlaxoSmithKline Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as Epelsiban ClinicalTrials.gov intervention name — accepted as the source's own label NCT02794467
3

NCT02257359

NCT02703181

NCT02213029

Known as EPELSIBAN BESYLATE ChEMBL registry synonym — accepted as the source's own label CHEMBL2037511
Known as GSK-557296B ChEMBL registry synonym — accepted as the source's own label CHEMBL2037511
Known as GSK557296 “Study IVF116828:A Multi-Cohort Phase I Study to Investigate the Pharmacokinetics, Pharmacodynamics and Tissue Concentrations of Epelsiban (GSK557296) in Healthy Female...” NCT02213029
4

“Epelsiban (GSK557296)” NCT02703181

NCT00549211

NCT01021553

NCT01669083

Action Inhibit “selective oxytocin receptor antagonist” PMID 23937679 Aug 2013
1

“Oxytocin receptor antagonist” CHEMBL2037511

Modality Small molecule CHEMBL2037511
Route Oral “Single and Repeat Oral Doses” NCT00549211
Target OXTR “Oxytocin receptor antagonist” CHEMBL2037511