Drugs / PF-00489791
last change Oct 2014 re-read 2 minutes ago

PF-00489791

also known as PF-489,791 · UK-489,791

Small molecule targets PDE5A via inhibition

Developed for
diabetic kidney disease · essential hypertension · postherpetic neuralgia · pulmonary arterial hypertension · Raynaud disease
Investigated by
Pfizer

Trials 6 · a red edge is where a trial was stopped

200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT02319148 Jul → Oct 2014 Pfizer Completed No outcome recorded
Phase 25 trials
Phase 2 NCT01200394 Dec 2010 → Jul 2013 diabetic kidney disease Pfizer Completed No outcome recorded
Phase 2 NCT01090492 Aug 2010 → May 2011 Raynaud disease Pfizer Completed No outcome recorded
Phase 2 NCT00853112 Apr 2009 → Jul 2010 pulmonary arterial hypertension Pfizer Terminated No outcome recorded
Phase 2 NCT00599638 Apr → Dec 2008 postherpetic neuralgia Pfizer Completed No outcome recorded
Phase 2 NCT00422461 Feb 2007 → Jan 2008 essential hypertension Pfizer Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as PF-00489791 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00422461
5

NCT00853112

NCT00599638

NCT01200394

NCT02319148

NCT01090492

Known as PF-489,791 ChEMBL registry synonym — accepted as the source's own label CHEMBL4210847
Known as UK-489,791 ChEMBL registry synonym — accepted as the source's own label CHEMBL4210847
Action Inhibit inhibitor of phosphodiesterase type 5” NCT01200394
1

“Phosphodiesterase 5A inhibitor” CHEMBL4210847

Modality Small molecule “a phosphodiesterase inhibitor” NCT01090492
Route Oral “PF-00489791 20 mg titrated to 40 mg, oral, tablets, once daily, for 28 days” NCT00422461
Target PDE5A “Phosphodiesterase 5A inhibitor” CHEMBL4210847