Drugs / M4344
last change May 2024 re-read 2 minutes ago

M4344

also known as gartisertib · VX-803

Small molecule targets ATR via inhibition

Developed for
breast cancer · cancer · ovarian carcinoma
Investigated by
EMD Serono Research & Development Institute, Inc. · Merck KGaA, Darmstadt, Germany · University of Alabama at Birmingham

Trials 3 · a red edge is where a trial was stopped

2015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT04149145 May 2023 → May 2024 ovarian carcinoma University of Alabama at Birmingham Withdrawn No outcome recorded
Phase 1 NCT02278250 Jan 2015 → Jun 2021 cancer EMD Serono Research & Development Institute, Inc. Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT04655183 Dec 2020 → Sep 2023 breast cancer EMD Serono Research & Development Institute, Inc. Withdrawn No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as M4344 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02278250
2

NCT04655183

NCT04149145

Known as gartisertib “A phase I study of ATR inhibitor gartisertib (M4344) as a single agent and in combination with carboplatin in patients with advanced solid tumours.” PMID 38287179 Jan 2024
Known as VX-803 ChEMBL registry synonym — accepted as the source's own label CHEMBL4650286
Action Inhibit “oral inhibitor of ataxia telangiectasia and Rad3-related protein (ATR)” PMID 38287179 Jan 2024
Modality Small molecule CHEMBL4650286
Route Oral “Participants received M4344 at a dose of 10 milligrams (mg) orally twice weekly (BIW)” NCT02278250
Target ATR “inhibitor of ataxia telangiectasia and Rad3-related protein (ATR)” PMID 38287179 Jan 2024