Drugs / Xentuzumab
last change May 2024 re-read 2 minutes ago

Xentuzumab

also known as BI 836845

Monoclonal antibody targets IGF1, IGF2, INSR via inhibition

Developed for
neoplasm · breast cancer · breast neoplasm · castration-resistant prostate carcinoma · non-small cell lung carcinoma · prostate cancer
Investigated by
Boehringer Ingelheim · Prostate Cancer UK · University of Oxford

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT05110495 Dec 2021 → Mar 2023 prostate cancer University of Oxford Completed No outcome recorded
Phase 17 trials
Phase 1 NCT03099174 May 2017 → May 2023 breast neoplasm Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02204072 Nov 2014 → Oct 2019 castration-resistant prostate carcinoma Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02191891 Oct 2014 → Apr 2018 non-small cell lung carcinoma Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02145741 Jun 2014 → Jul 2015 neoplasm Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02123823 May 2014 → Nov 2016 neoplasm Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT01403974 Jul 2011 → Jul 2015 neoplasm Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT01317420 Apr 2011 → Feb 2016 neoplasm Boehringer Ingelheim Completed No outcome recorded
Phase 21 trial
Phase 2 NCT03659136 Nov 2018 → Aug 2021 breast cancer Boehringer Ingelheim Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 13 sources stand behind the page.

FieldValueCited text
Known as xentuzumab xentuzumab (BI 836845) 1000 mg + everolimus 10 mg + exemestane 25 mg - Phase II” NCT02123823
5

NCT02191891

NCT05110495

NCT02145741

NCT03659136

NCT03099174

Known as BI 836845 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01317420
3

NCT02123823

NCT02204072

NCT01403974

Action Inhibit “Xentuzumab, an insulin-like growth factor (IGF)-1/IGF-2-neutralising antibody, binds IGF-1 and IGF-2, inhibiting their growth-promoting signalling.” PMID 32161368 Mar 2020
2

“Insulin-like growth factor II inhibitor” CHEMBL4297850

“Insulin-like growth factor I inhibitor” CHEMBL4297850

Modality Monoclonal antibody “Xentuzumab is a humanised monoclonal antibodyPMID 37308971 Jun 2023
Route Intravenous “Patients received xentuzumab intravenously at a starting dose of 750 mg/wk.” PMID 34870878 Jan 2022
Target IGF1 “Insulin-like growth factor I inhibitor” CHEMBL4297850
Target IGF2 “Insulin-like growth factor II inhibitor” CHEMBL4297850
Target INSR “neutralises the IGF ligands to inhibit activation of IGF-1R and INSR-A” NCT05110495