Drugs / Verinurad
last change Apr 2022 re-read 2 minutes ago

Verinurad

also known as RDEA3170

Small molecule targets SLC22A12 via inhibition

Developed for
gout · chronic kidney disease · diastolic heart failure · proteinuria · type 2 diabetes mellitus
Investigated by
Ardea Biosciences, Inc. · AstraZeneca · Parexel

Trials 21 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 113 trials
Phase 1 NCT04550234 Apr → Jul 2021 chronic kidney disease AstraZeneca Completed No outcome recorded
Phase 1 NCT04532918 Sep → Nov 2020 chronic kidney disease AstraZeneca Completed No outcome recorded
Phase 1 NCT04256629 Mar → Aug 2020 AstraZeneca Completed No outcome recorded
Phase 1 NCT04024501 Jul → Sep 2019 chronic kidney disease AstraZeneca Completed No outcome recorded
Phase 1 NCT03836599 Jan → Apr 2019 chronic kidney disease AstraZeneca Completed No outcome recorded
Phase 1 NCT02608710 Nov → Dec 2015 gout Ardea Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02448368 May → Jun 2015 Ardea Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02279641 Nov 2014 → Apr 2015 gout Ardea Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02336594 Nov 2014 → Jan 2015 gout Ardea Biosciences, Inc. Completed No outcome recorded
Phase 1 NCT02219516 Aug 2014 → Oct 2015 gout Ardea Biosciences, Inc. Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02317861 Dec 2014 → Jun 2015 gout AstraZeneca Completed No outcome recorded
Phase 27 trials
Phase 2 NCT04327024 May 2020 → Apr 2022 diastolic heart failure AstraZeneca Completed No outcome recorded
Phase 2 NCT03990363 Jul 2019 → Nov 2021 chronic kidney disease AstraZeneca Completed No outcome recorded
Phase 2 NCT03118739 May 2017 → Aug 2018 proteinuria, type 2 diabetes mellitus AstraZeneca Completed No outcome recorded
Phase 2 NCT02498652 Jul → Nov 2015 gout Ardea Biosciences, Inc. Completed No outcome recorded
Phase 2 NCT02246673 Oct 2014 → Jul 2015 gout Ardea Biosciences, Inc. Completed No outcome recorded
Phase 2 NCT02078219 Jan 2014 → Mar 2015 gout AstraZeneca Completed No outcome recorded
Phase 2 NCT01927198 Aug 2013 → May 2014 gout Ardea Biosciences, Inc. Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT03316131 Background Oct 2017 → Jul 2018 AstraZeneca Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 24 sources stand behind the page.

FieldValueCited text
Known as Verinurad Verinurad (RDEA3170) is a high affinity, selective uric acid transporter (URAT1) inhibitor indevelopment for treating gout and asymptomatic hyperuricaemia.” PMID 29531784 Feb 2018
12

Verinurad (RDEA3170) is a high-affinity inhibitor of the URAT1 transporter in clinical development for treating gout and asymptomatic hyperuricaemia.” PMID 29868853 Sep 2018

Verinurad (RDEA3170) is a high-affinity, selective URAT1 transporter inhibitor in development for treating gout and asymptomatic hyperuricemia.” PMID 29949102 Aug 2018

“Randomized patients will receive orally once daily fixed dose of verinurad in 2 treatment sequences AB or BA for 7 consecutive days.” NCT03316131

Verinurad (RDEA3170) is a high-affinity, selective URAT1 inhibitor in development for treating gout and asymptomatic hyperuricaemia.” PMID 29657831 Apr 2018

NCT04532918

NCT04327024

NCT03990363

NCT03118739

NCT04256629

NCT03836599

NCT04024501

NCT04550234

Known as RDEA3170 “Verinurad (RDEA3170) is a high affinity, selective uric acid transporter (URAT1) inhibitor indevelopment for treating gout and asymptomatic hyperuricaemia.” PMID 29531784 Feb 2018
13

“Verinurad (RDEA3170) is a high-affinity inhibitor of the URAT1 transporter in clinical development for treating gout and asymptomatic hyperuricaemia.” PMID 29868853 Sep 2018

“Verinurad (RDEA3170) is a high-affinity, selective URAT1 inhibitor in development for treating gout and asymptomatic hyperuricaemia.” PMID 29657831 Apr 2018

“Verinurad (RDEA3170) is a novel URAT1 inhibitor in Phase 2 development for chronic kidney disease and heart failure.” NCT03990363

NCT02336594

NCT01927198

NCT02219516

NCT02608710

NCT02078219

NCT01910506

NCT01872832

NCT02448368

NCT01883167

NCT02279641

Action Inhibit “Solute carrier family 22 member 12 inhibitor” CHEMBL3707347
1

“the investigational URAT1 inhibitor RDEA3170” NCT01883167

Modality Small molecule CHEMBL3707347
Route Oral “RDEA3170 oral solution” NCT01910506
Target SLC22A12 “Solute carrier family 22 member 12 inhibitor” CHEMBL3707347