Drugs / ASTX727 Dose Escalation
last change Dec 2019 re-read 2 minutes ago

ASTX727 Dose Escalation

Small molecule targets DNMT1 via inhibition

Developed for
myelodysplastic syndrome
Investigated by
Astex Pharmaceuticals, Inc.

Trials 1 · a red edge is where a trial was stopped

2015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/2 NCT02103478 Oct 2014 → Jun 2018 myelodysplastic syndrome Astex Pharmaceuticals, Inc. Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 2 sources stand behind the page.

FieldValueCited text
Known as ASTX727 Dose Escalation ClinicalTrials.gov intervention name — accepted as the source's own label NCT02103478
Action Inhibit “Decitabine, a DNA methyltransferase 1 inhibitor or DNA hypomethylating compound” PMID 30926081 Apr 2019
Modality Small molecule “Decitabine, a DNA methyltransferase 1 inhibitor or DNA hypomethylating compound, is not readily orally bioavailable” PMID 30926081 Apr 2019
Route Oral oral decitabine and cedazuridine were given on days 1-5” PMID 30926081 Apr 2019
Target DNMT1 “Decitabine, a DNA methyltransferase 1 inhibitor or DNA hypomethylating compound” PMID 30926081 Apr 2019