Drugs / KTX-1001
last change Feb 2023 re-read 2 minutes ago

KTX-1001

Small molecule targets NSD2 via inhibition

Developed for
plasma cell myeloma
Investigated by
Bristol-Myers Squibb · K36 Therapeutics, Inc.

Trials 1 · a red edge is where a trial was stopped

202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT05651932 Feb 2023 → Dec 2027 expected plasma cell myeloma K36 Therapeutics, Inc. Recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 1 source stands behind the page.

FieldValueCited text
Known as KTX-1001 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05651932
Action Inhibit “small molecule inhibitor of the histone lysine methyl transferase MMSET” NCT05651932
Modality Small molecule “a novel, orally available, selective, and potent small molecule inhibitor of the histone lysine methyl transferase MMSET” NCT05651932
Route Oral “KTX-1001: Orally for 28 days each cycle until progression” NCT05651932
Target NSD2 “inhibitor of the histone lysine methyl transferase MMSET (also known as NSD2/WHSC1)” NCT05651932