Drugs / KTX-1001
last change Feb 2023 re-read 9 days ago

KTX-1001

Small molecule targets NSD2 via inhibition

Developed for
plasma cell myeloma
Investigated by
Bristol-Myers Squibb · K36 Therapeutics, Inc.

Trials 1

202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT05651932 Feb 2023 → Dec 2027 expected plasma cell myeloma K36 Therapeutics, Inc. Recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 1 source stands behind the page.

FieldValueCited text
Known as KTX-1001 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05651932 ↗
Action Inhibit “small molecule inhibitor of the histone lysine methyl transferase MMSET” NCT05651932 ↗
Modality Small molecule “a novel, orally available, selective, and potent small molecule inhibitor of the histone lysine methyl transferase MMSET” NCT05651932 ↗
Route Oral “KTX-1001: Orally for 28 days each cycle until progression” NCT05651932 ↗
Target NSD2 “inhibitor of the histone lysine methyl transferase MMSET (also known as NSD2/WHSC1)” NCT05651932 ↗