Drugs / Cebranopadol
last change Jan 2025 re-read 2 minutes ago

Cebranopadol

also known as GRT6005

Small molecule targets OPRL1 via activation

Developed for
chronic pain syndrome · neoplasm · diabetic neuropathy · diabetic polyneuropathy · osteoarthritis, knee
Investigated by
Tris Pharma, Inc. · Forest Laboratories · National Institutes of Health (NIH)

Trials 16 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT06453265 Jun → Nov 2024 substance abuse Tris Pharma, Inc. Completed No outcome recorded
Phase 1 NCT05491785 Jul 2022 → Mar 2023 Tris Pharma, Inc. Completed No outcome recorded
Phase 1 NCT05256108 Mar → Jul 2022 substance abuse Tris Pharma, Inc. Completed No outcome recorded
Phase 1 NCT03958123 Jul → Nov 2013 Tris Pharma, Inc. Completed No outcome recorded
Phase 1 NCT03882762 Jun 2013 → Sep 2014 Tris Pharma, Inc. Completed No outcome recorded
Phase 1 NCT03757559 Apr 2013 → Mar 2014 substance abuse Tris Pharma, Inc. Completed No outcome recorded
Phase 26 trials
Phase 2 NCT01939366 Sep 2013 → Jan 2015 chronic pain syndrome, diabetes mellitus, diabetic neuropathy Tris Pharma, Inc. Completed No outcome recorded
Phase 2 NCT01709214 Dec 2012 → Apr 2014 Tris Pharma, Inc. Completed No outcome recorded
Phase 2 NCT01725087 Nov 2012 → Jul 2014 Tris Pharma, Inc. Completed No outcome recorded
Phase 2 NCT01357837 May → Dec 2011 osteoarthritis, knee Tris Pharma, Inc. Completed No outcome recorded
Phase 2 NCT00878293 Apr 2009 → May 2010 diabetic polyneuropathy Tris Pharma, Inc. Completed No outcome recorded
Phase 2 NCT00872885 Mar → Aug 2009 Tris Pharma, Inc. Completed No outcome recorded
Phase 34 trials
Phase 3 NCT06545097 Sep → Dec 2024 Tris Pharma, Inc. Completed No outcome recorded
Phase 3 NCT06423703 Jul 2024 → Jan 2025 Tris Pharma, Inc. Completed No outcome recorded
Phase 3 NCT02031432 Dec 2013 → Apr 2016 chronic pain syndrome, neoplasm Tris Pharma, Inc. Completed No outcome recorded
Phase 3 NCT01964378 Oct 2013 → Oct 2015 chronic pain syndrome, neoplasm Tris Pharma, Inc. Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01347671 Comparator May 2011 → Jan 2012 diabetic polyneuropathy Tris Pharma, Inc. Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 19 sources stand behind the page.

FieldValueCited text
Known as Cebranopadol ClinicalTrials.gov intervention name — accepted as the source's own label NCT06545097
11

NCT03882762

NCT01964378

NCT01939366

NCT01709214

NCT05491785

NCT06423703

NCT03757559

NCT06453265

NCT02031432

NCT03958123

NCT05256108

Known as GRT6005 “The objective of this study was to evaluate the pharmacokinetics (PK), safety and tolerability profile of cebranopadol (GRT6005) in patients with varying degree of renal...” NCT03882762
8

“The objective of this study was to evaluate the effects of cebranopadol (GRT6005) on the electrical activity of the heart in healthy participants.” NCT03958123

“The primary objective of this study was to evaluate the abuse potential of single doses of cebranopadol (GRT6005) relative to hydromorphone” NCT03757559

“Cebranopadol (GRT6005) Low-Dose Range” NCT01709214

NCT01725087

NCT00872885

NCT00878293

NCT01347671

NCT01357837

Action Activate “opioid peptide receptor agonism” PMID 30365202 Jan 2019
1

“Nociceptin receptor agonist” CHEMBL2364605

Modality Small molecule CHEMBL2364605
Route Oral “liquid formulation for oral application” NCT00878293
Target OPRL1 “Nociceptin receptor agonist” CHEMBL2364605