Drugs / RAVOXERTINIB
last change Dec 2016 re-read 2 minutes ago

RAVOXERTINIB

also known as GDC-0994 · RG-7842

Small molecule targets MAPK1, MAPK3 via inhibition

Developed for
cancer · colorectal cancer · metastatic melanoma · non-small cell lung carcinoma
Investigated by
Genentech, Inc.

Trials 2 · a red edge is where a trial was stopped

20142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT02457793 Jun 2015 → Dec 2016 colorectal cancer, metastatic melanoma, non-small cell lung carcinoma Genentech, Inc. Completed No outcome recorded
Phase 1 NCT01875705 Jun 2013 → Sep 2016 cancer Genentech, Inc. Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 3 sources stand behind the page.

FieldValueCited text
Known as RAVOXERTINIB ChEMBL registry synonym — accepted as the source's own label CHEMBL3544964
Known as GDC-0994 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01875705
1

NCT02457793

Known as RG-7842 ChEMBL registry synonym — accepted as the source's own label CHEMBL3544964
Action Inhibit “MAP kinase ERK2 inhibitor” CHEMBL3544964
1

“MAP kinase ERK1 inhibitor” CHEMBL3544964

Modality Small molecule CHEMBL3544964
Route Oral oral dosing of cobimetinib and GDC-0994 administered in combination” NCT02457793
Target MAPK1 “MAP kinase ERK2 inhibitor” CHEMBL3544964
Target MAPK3 “MAP kinase ERK1 inhibitor” CHEMBL3544964