Drugs / Icenticaftor
last change Aug 2023 re-read 2 minutes ago

Icenticaftor

English name icenticaftor
also known as QBW251

Small molecule targets CFTR

Developed for
chronic obstructive pulmonary disease · bronchiectasis · cystic fibrosis
Investigated by
Novartis Pharmaceuticals · Innovative Medicines Initiative

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT04587622 Oct 2020 → Sep 2022 liver failure Novartis Pharmaceuticals Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02190604 Jul 2012 → Nov 2015 cystic fibrosis Novartis Pharmaceuticals Terminated No outcome recorded
Phase 24 trials
Phase 2 NCT04396366 Feb 2021 → Jun 2023 bronchiectasis Novartis Pharmaceuticals Terminated No outcome recorded
Phase 2 NCT04268823 Sep 2020 → Sep 2022 chronic obstructive pulmonary disease Novartis Pharmaceuticals Terminated No outcome recorded
Phase 2 NCT04072887 Sep 2019 → Oct 2021 chronic obstructive pulmonary disease Novartis Pharmaceuticals Completed No outcome recorded
Phase 2 NCT02449018 Apr 2015 → Dec 2016 chronic obstructive pulmonary disease Novartis Pharmaceuticals Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as icenticaftor “The aim of this phase IIb dose-finding study was to compare a CFTR potentiator, icenticaftor (QBW251), with placebo in patients with COPD and chronic bronchitis.” PMID 37411039 Aug 2023
1

NCT04587622

Known as QBW251 “The aim of this phase IIb dose-finding study was to compare a CFTR potentiator, icenticaftor (QBW251), with placebo in patients with COPD and chronic bronchitis.” PMID 37411039 Aug 2023
5

“Single oral dose of 300 mg of icenticaftor (QBW251)” NCT04587622

NCT02449018

NCT04268823

NCT04396366

NCT02190604

Action Activate “an oral potentiator of the cystic fibrosis (CF) transmembrane conductance regulator (CFTR) channel” PMID 33293212 Dec 2020
Modality Small molecule CHEMBL4650318
Route Oral “Capsule - oral dose” NCT02190604
Target CFTR “an oral potentiator of the cystic fibrosis (CF) transmembrane conductance regulator (CFTR) channel” PMID 33293212 Dec 2020