Drugs / DBPR108
last change Jun 2025 re-read 2 minutes ago

DBPR108

also known as prusogliptin

Small molecule targets DPP4 via inhibition

Developed for
type 2 diabetes mellitus
Investigated by
CSPC ZhongQi Pharmaceutical Technology Co., Ltd. · National Health Research Institutes, Taiwan · CSPC Ouyi Pharmaceutical Co., Ltd.

Trials 13 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 19 trials
Phase 1 NCT05150626 May → Jun 2022 CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT05146869 Dec 2021 → Mar 2022 type 2 diabetes mellitus CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT05072028 Nov 2021 CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT05045313 Oct → Dec 2021 CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT04859439 Jun → Nov 2021 impaired renal function disease CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT04859426 Jun 2021 → May 2022 CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT04859452 May → Jul 2021 CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 1 NCT02163278 Jun 2014 → Jan 2015 type 2 diabetes mellitus National Health Research Institutes, Taiwan Completed No outcome recorded
Phase 1 NCT01650324 Jul → Dec 2012 type 2 diabetes mellitus National Health Research Institutes, Taiwan Completed No outcome recorded
Phase 21 trial
Phase 2 NCT04124484 Oct 2017 → Feb 2019 type 2 diabetes mellitus CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 33 trials
Phase 3 NCT07026968 Jun 2025 → Oct 2026 expected type 2 diabetes mellitus CSPC Ouyi Pharmaceutical Co., Ltd. Active not recruiting No outcome recorded
Phase 3 NCT04218734 Jan 2020 → Jun 2021 type 2 diabetes mellitus CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded
Phase 3 NCT04161430 Jan 2020 → Jun 2022 type 2 diabetes mellitus CSPC ZhongQi Pharmaceutical Technology Co., Ltd. Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 15 sources stand behind the page.

FieldValueCited text
Known as DBPR108 DBPR108NCT05045313
12

NCT04859426

NCT05150626

NCT04859452

NCT05045313

NCT04859439

NCT05072028

NCT04161430

NCT04218734

NCT01650324

NCT04124484

NCT05146869

NCT02163278

Known as prusogliptin “DBPR108 (prusogliptin) is a novel, orally bioavailable dipeptidyl peptidase-4 (DPP-4) inhibitor.” PMID 40252162 Apr 2025
1

NCT07026968

Action Inhibit “dipeptidyl peptidase 4 (DPP4) inhibitor DBPR108” NCT01650324
Modality Small molecule CHEMBL1082462
Route Oral “single oral doses of DBPR108 in healthy male subjects” NCT01650324
Target DPP4 DPP4 inhibitor DBPR108” NCT02163278