Drugs / Fasiglifam
last change Jan 2016 re-read 2 minutes ago

Fasiglifam

English name fasiglifam
also known as TAK-875 · AK875 · CPD 9A · TAK-875 ANHYDROUS

Small molecule targets FFAR1 via activation

Developed for
type 2 diabetes mellitus · diabetes mellitus · cardiovascular disorder · glucose metabolism disease
Investigated by
Takeda

Trials 18 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01496443 Jan → May 2012 Takeda Completed No outcome recorded
Phase 1 NCT00949091 Jan → Jul 2009 type 2 diabetes mellitus Takeda Completed No outcome recorded
Phase 23 trials
Phase 2 NCT01982253 Oct 2013 → Jan 2014 type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 2 NCT01414920 Aug 2011 → Aug 2012 type 2 diabetes mellitus Takeda Completed No outcome recorded
Phase 2 NCT01007097 Dec 2009 → Sep 2010 type 2 diabetes mellitus Takeda Completed No outcome recorded
Phase 313 trials
Phase 3 NCT02015780 Dec 2013 → Jan 2016 chronic kidney disease, type 2 diabetes mellitus Takeda Withdrawn No outcome recorded
Phase 3 NCT01834274 Jun 2013 → Mar 2014 type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 3 NCT01829464 May 2013 → Feb 2014 type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 3 NCT01829477 Apr 2013 → Feb 2014 type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 3 NCT01647542 Oct 2012 → Feb 2014 type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 3 NCT01609582 Jun 2012 → May 2014 cardiovascular disorder, type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 3 NCT01585792 May → Dec 2012 Takeda Completed No outcome recorded
Phase 3 NCT01549964 Apr 2012 → Mar 2014 glucose metabolism disease Takeda Terminated No outcome recorded
Phase 3 NCT01481116 Jan 2012 → Mar 2014 type 2 diabetes mellitus Takeda Terminated No outcome recorded
Phase 3 NCT01433419 Jan → Dec 2012 diabetes mellitus Takeda Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 20 sources stand behind the page.

FieldValueCited text
Known as fasiglifam “Due to potential concerns about liver safety, on balance, the benefits of treating patients with fasiglifam (TAK-875) do not outweigh the potential risks.” NCT01647542
8

“Due to potential concerns about liver safety, on balance, the benefits of treating patients with fasiglifam (TAK-875) do not outweigh the potential risks.” NCT01481116

“Due to potential concerns about liver safety, on balance, the benefits of treating patients with fasiglifam (TAK-875) do not outweigh the potential risks.” NCT01829477

“The drug being tested in this study is called TAK-875 (fasiglifam).” NCT01829464

NCT01456195

NCT02015780

NCT01982253

NCT01834274

NCT01549964

Known as AK875 ChEMBL registry synonym — accepted as the source's own label CHEMBL1829174
Known as CPD 9A ChEMBL registry synonym — accepted as the source's own label CHEMBL1829174
Known as TAK-875 “The purpose of this study is to determine the efficacy and safety of TAK-875 (fasiglifam), once daily (QD), in participants with type 2 diabetes mellitus (T2DM).” NCT01456195
15

TAK-875 is under clinical development for the treatment of type 2 diabetes mellitus in humans.” NCT01007097

“Fasiglifam (TAK-875) tablets” NCT01834274

“Fasiglifam (TAK-875) tablets” NCT01549964

NCT01414920

NCT01829477

NCT01829464

NCT01481116

NCT01433419

NCT00949091

NCT01585792

NCT01433406

NCT01496443

NCT01647542

NCT01609582

NCT01433393

Known as TAK-875 ANHYDROUS ChEMBL registry synonym — accepted as the source's own label CHEMBL1829174
Action Activate “selective pharmacological activation of this receptor by TAK-875” PMID 22374408 Feb 2012
1

“Free fatty acid receptor 1 positive allosteric modulator” CHEMBL1829174

Modality Small molecule CHEMBL1829174
Route Oral “TAK-875 25 mg tablets, orally” NCT00949091
Target FFAR1 “Free fatty acid receptor 1 positive allosteric modulator” CHEMBL1829174