Drugs / E7386
last change Jun 2026 re-read 2 minutes ago

E7386

Small molecule

Developed for
colorectal neoplasm · hepatocellular carcinoma · colorectal cancer · endometrial cancer · melanoma · neoplasm
Investigated by
Eisai Inc. · Merck Sharp & Dohme LLC

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT05607537 Oct 2022 → Aug 2023 Eisai Inc. Completed No outcome recorded
Phase 1 NCT04840927 Apr 2021 → May 2023 Eisai Inc. Withdrawn No outcome recorded
Phase 1 NCT03996226 Jun → Oct 2019 Eisai Inc. Completed No outcome recorded
Phase 1 NCT03833700 Mar 2019 → Mar 2027 expected colorectal neoplasm Eisai Inc. Active not recruiting No outcome recorded
Phase 1 NCT03264664 Jul 2017 → Mar 2027 expected neoplasm Eisai Inc. Active not recruiting No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT05091346 Oct 2021 → Oct 2024 colorectal neoplasm, hepatocellular carcinoma, melanoma Eisai Inc. Completed No outcome recorded
Phase 1/2 NCT04008797 Jul 2019 → Mar 2027 expected colorectal cancer, endometrial cancer, hepatocellular carcinoma Eisai Inc. Active not recruiting No outcome recorded

Evidence & citations 4 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as E7386 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05607537
6

NCT03833700

NCT05091346

NCT04840927

NCT04008797

NCT03996226

NCT03264664

Action Inhibit “BACKGROUND: We present data from the Phase 1 open-label Study 101 of E7386, an oral protein-protein interaction inhibitor reported to block the CBP/β-catenin interaction, in...” PMID 42243349 Jun 2026
Modality Small molecule “E7386, a novel small-molecule inhibitor, has been shown to enhance anti-angiogenesis when combined with lenvatinib.” PMID 40318924 Apr 2025
Route Oral “E7386 will be administered as a single agent orally” NCT03264664