Drugs / Iruplinalkib
last change Jan 2026 re-read 2 minutes ago

Iruplinalkib

also known as WX-0593

targets ALK, ROS1 via inhibition

Developed for
non-small cell lung carcinoma
Investigated by
Qilu Pharmaceutical Co., Ltd. · Henan Cancer Hospital · Shanghai Pulmonary Hospital, Shanghai, China · Tianjin Medical University Cancer Institute and Hospital

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT06436885 Feb 2024 → Dec 2025 non-small cell lung carcinoma Henan Cancer Hospital Unknown No outcome recorded
Phase 11 trial
Phase 1 NCT05716126 Apr → Dec 2020 Qilu Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 23 trials
Phase 2 NCT07330076 Jan 2026 → Dec 2030 expected non-small cell lung carcinoma Tianjin Medical University Cancer Institute and Hospital Not yet recruiting No outcome recorded
Phase 2 NCT06282536 Mar 2024 → Jun 2025 overdue Shanghai Pulmonary Hospital, Shanghai, China Not yet recruiting No outcome recorded
Phase 2 NCT04641754 Mar 2019 → Dec 2020 non-small cell lung carcinoma Qilu Pharmaceutical Co., Ltd. Unknown No outcome recorded
Phase 31 trial
Phase 3 NCT04632758 Jun 2019 → Dec 2024 non-small cell lung carcinoma Qilu Pharmaceutical Co., Ltd. Unknown No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as Iruplinalkib Iruplinalkib (WX-0593) is a new-generation, potent ALK tyrosine kinase inhibitor (TKI) that has been found to have systemic and central nervous system (CNS) efficacy in...” PMID 38280448 Jan 2024
5

“Efficacy and safety of iruplinalkib (WX-0593) in ALK-positive crizotinib-resistant advanced non-small cell lung cancer patients: a single-arm, multicenter phase II study (INTELLECT).” PMID 36829154 Feb 2023

NCT07330076

NCT06282536

NCT06436885

NCT05716126

Known as WX-0593 “Iruplinalkib (WX-0593) is a new-generation, potent ALK tyrosine kinase inhibitor (TKI) that has been found to have systemic and central nervous system (CNS) efficacy in...” PMID 38280448 Jan 2024
2

“Iruplinalkib (WX-0593) is an anaplastic lymphoma kinase (ALK)/c-ros oncogene 1 (ROS1) tyrosine kinase inhibitor.” PMID 36829154 Feb 2023

“Volunteer will receive a single oral dose of 120 mg \[14C\]Iruplinalkib (WX-0593) as a solution on Day 1” NCT05716126

Action Inhibit “potent ALK tyrosine kinase inhibitor (TKI)” PMID 38280448 Jan 2024
Route Oral “Patients received iruplinalkib 180 mg orally once daily for a 21-day cycle with a 7-day lead-in phase at 60 mg orally once daily.” PMID 36829154 Feb 2023
Target ALK “potent ALK tyrosine kinase inhibitor (TKI)” PMID 38280448 Jan 2024