Drugs / Icrucumab
last change Jul 2017 re-read 2 minutes ago

Icrucumab

also known as ICR · IMC-18F1

Monoclonal antibody targets FLT1 via inhibition

Developed for
breast cancer · cancer · carcinoma of urethra · colon carcinoma · rectal carcinoma · renal pelvis carcinoma · ureter carcinoma · urothelial carcinoma
Investigated by
Eli Lilly and Company

Trials 4 · a red edge is where a trial was stopped

2006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT00782002 Jul 2006 → Mar 2009 cancer Eli Lilly and Company Completed No outcome recorded
Phase 23 trials
Phase 2 NCT01282463 Apr 2011 → Feb 2015 carcinoma of urethra, renal pelvis carcinoma, ureter carcinoma, urothelial carcinoma Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT01234402 Mar 2011 → Oct 2013 breast cancer Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT01111604 Aug 2010 → Dec 2013 colon carcinoma, rectal carcinoma Eli Lilly and Company Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as icrucumab Icrucumab (ICR) and ramucirumab (RAM) bind vascular endothelial growth factor (VEGF) receptors 1 and 2 (VEGFR-1 and -2), respectively.” PMID 28220020 Feb 2017
3

“IMC-18F1 (icrucumab), a human monoclonal antibody against vascular endothelial growth factor receptor-1 (VEGFR-1)” PMID 23903897 Aug 2013

NCT01111604

NCT01282463

Known as ICR Icrucumab (ICR) and ramucirumab (RAM) bind vascular endothelial growth factor (VEGF) receptors 1 and 2 (VEGFR-1 and -2), respectively.” PMID 28220020 Feb 2017
Known as IMC-18F1 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00782002
Action Inhibit “potently inhibits ligand-dependent phosphorylation of VEGFR-1 and downstream signaling” PMID 23903897 Aug 2013
1

“Vascular endothelial growth factor receptor 1 antagonist” CHEMBL1743030

Modality Monoclonal antibody “a human monoclonal antibody against vascular endothelial growth factor receptor-1 (VEGFR-1)” PMID 23903897 Aug 2013
Route Intravenous “12 mg/kg IV, days 1 and 8” PMID 28220020 Feb 2017
Target FLT1 “Vascular endothelial growth factor receptor 1 antagonist” CHEMBL1743030