Drugs / Acumapimod
last change Nov 2019 re-read 2 minutes ago

Acumapimod

also known as BCT197

Small molecule targets MAPK14 via inhibition

Developed for
chronic obstructive pulmonary disease · acute kidney injury
Investigated by
Mereo BioPharma · Novartis

Trials 5 · a red edge is where a trial was stopped

20112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT03498170 Mar → May 2018 Mereo BioPharma Completed No outcome recorded
Phase 1 NCT02926326 Sep → Oct 2016 Mereo BioPharma Completed No outcome recorded
Phase 23 trials
Phase 2 NCT02700919 Aug 2016 → Nov 2017 chronic obstructive pulmonary disease Mereo BioPharma Completed No outcome recorded
Phase 2 NCT01336959 Sep 2011 → Nov 2013 acute kidney injury Mereo BioPharma Terminated No outcome recorded
Phase 2 NCT01332097 Mar 2011 → May 2013 chronic obstructive pulmonary disease Mereo BioPharma Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as Acumapimod Acumapimod is a potent, selective, oral, p38 inhibitor under investigation for treatment of acute exacerbations of COPD (AECOPD).” PMID 31682162 Nov 2019
Known as BCT197 “Phase II Study of Single/Repeated Doses of Acumapimod (BCT197) to Treat Acute Exacerbations of COPD.” PMID 31682162 Nov 2019
4

NCT03498170

NCT02700919

NCT01336959

NCT02926326

Action Inhibit “Acumapimod is a potent, selective, oral, p38 inhibitor under investigation for treatment of acute exacerbations of COPD (AECOPD).” PMID 31682162 Nov 2019
1

“MAP kinase p38 alpha inhibitor” CHEMBL5314397

Modality Small molecule CHEMBL5314397
Route Oral “Acumapimod is a potent, selective, oral, p38 inhibitor under investigation for treatment of acute exacerbations of COPD (AECOPD).” PMID 31682162 Nov 2019
Target MAPK14 “MAP kinase p38 alpha inhibitor” CHEMBL5314397