Drugs / Tabalumab
last change Nov 2015 re-read 2 minutes ago

Tabalumab

English name tabalumab
also known as LY2127399

Monoclonal antibody targets TNFSF13B via inhibition

Developed for
rheumatoid arthritis · systemic lupus erythematosus · plasma cell myeloma · chronic renal failure syndrome · relapsing-remitting multiple sclerosis
Investigated by
Eli Lilly and Company · Applied Molecular Evolution

Trials 21 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT01556438 Jul 2012 → Feb 2015 plasma cell myeloma Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01253291 May 2010 → Sep 2013 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01253226 Sep 2009 → Aug 2011 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT00689507 Mar 2008 → Jan 2013 plasma cell myeloma Applied Molecular Evolution Completed No outcome recorded
Phase 28 trials
Phase 2 NCT01602224 Jul 2012 → Jul 2014 plasma cell myeloma Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT01576549 May 2012 → May 2013 rheumatoid arthritis Eli Lilly and Company Terminated No outcome recorded
Phase 2 NCT01200290 Apr 2011 → Mar 2014 chronic renal failure syndrome Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00882999 Apr 2009 → Feb 2011 relapsing-remitting multiple sclerosis Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00837811 Feb 2009 → Jan 2011 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00785928 Oct 2008 → Jan 2010 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00689728 Jun 2008 → Feb 2010 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00308282 Mar 2006 → Jun 2007 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 39 trials
Phase 3 NCT02041091 Jan → Oct 2014 systemic lupus erythematosus Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT01676701 Sep 2012 → Aug 2013 rheumatoid arthritis Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT01488708 Jan 2012 → Oct 2015 systemic lupus erythematosus Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT01215942 Jun 2011 → Feb 2014 rheumatoid arthritis Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT01205438 Jan 2011 → Aug 2014 systemic lupus erythematosus Eli Lilly and Company Completed No outcome recorded
Phase 3 NCT01202773 Jan 2011 → Mar 2013 rheumatoid arthritis Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT01202760 Jan 2011 → Dec 2012 rheumatoid arthritis Eli Lilly and Company Completed No outcome recorded
Phase 3 NCT01196091 Dec 2010 → Jul 2014 systemic lupus erythematosus Eli Lilly and Company Completed No outcome recorded
Phase 3 NCT01198002 Dec 2010 → Dec 2012 rheumatoid arthritis Eli Lilly and Company Terminated No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 24 sources stand behind the page.

FieldValueCited text
Known as tabalumab “To assess the dose-response relationship, efficacy and safety of tabalumab, a human monoclonal antibody that neutralises membrane-bound and soluble B-cell activating factor...” PMID 23599435 Apr 2013
8

“Efficacy and safety of tabalumab, an anti-B-cell-activating factor monoclonal antibody, in patients with rheumatoid arthritis who had an inadequate response to methotrexate...” PMID 25873635 Apr 2015

“A 52-week, open-label study evaluating the safety and efficacy of tabalumab, an anti-B-cell-activating factor monoclonal antibody, for rheumatoid arthritis.” PMID 25168268 Aug 2014

“OBJECTIVE: Tabalumab, a fully human IgG4 monoclonal antibody, neutralizes soluble and membrane-bound BAFF.” PMID 23359344 Apr 2013

“LY2127399 (Tabalumab)” NCT01253226

NCT01676701

NCT01602224

NCT02041091

NCT01556438

Known as LY2127399 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00689507
15

NCT00308282

NCT01205438

NCT00837811

NCT01253291

NCT01198002

NCT01488708

NCT01253226

NCT00689728

NCT01215942

NCT01196091

NCT01576549

NCT01200290

NCT01202773

NCT01202760

NCT00882999

Action Inhibit “neutralizes soluble and membrane-bound BAFF” PMID 23359344 Apr 2013
Modality Monoclonal antibody “a fully human IgG4 monoclonal antibodyPMID 23359344 Apr 2013
Route Intravenous “30 mg, 60 mg or 160 mg, IV (in the vein) in weeks 0, 3 and 6” NCT00308282
Target TNFSF13B “neutralizes soluble and membrane-bound BAFF” PMID 23359344 Apr 2013