Drugs / BI 187004
last change Aug 2021 re-read 2 minutes ago

BI 187004

Small molecule targets HSD11B1 via inhibition

Developed for
type 2 diabetes mellitus
Investigated by
Boehringer Ingelheim

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT02305901 Dec 2014 → Mar 2015 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02254148 Oct → Dec 2014 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02161432 Jun → Sep 2014 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02109679 May → Jul 2014 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT01874483 Jun → Dec 2013 type 2 diabetes mellitus Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT01587417 Apr → Oct 2012 Boehringer Ingelheim Completed No outcome recorded
Phase 21 trial
Phase 2 NCT02150824 Jul 2014 → Jul 2015 type 2 diabetes mellitus Boehringer Ingelheim Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as BI 187004 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02150824
6

NCT01587417

NCT02161432

NCT01874483

NCT02109679

NCT02254148

NCT02305901

Action Inhibit “BI 187004, an inhibitor of 11beta-hydroxysteroid dehydrogenase-1” PMID 34391480 Aug 2021
1

“11-beta-hydroxysteroid dehydrogenase 1 inhibitor” CHEMBL3669417

Modality Small molecule CHEMBL3669417
Route Oral “single oral doses of BI 187004” PMID 34391480 Aug 2021
Target HSD11B1 “11-beta-hydroxysteroid dehydrogenase 1 inhibitor” CHEMBL3669417