Drugs / SRT2104
last change Mar 2013 re-read 2 minutes ago

SRT2104

Small molecule targets SIRT1 via activation

Developed for
type 2 diabetes mellitus · ulcerative colitis · muscular atrophy · psoriasis
Investigated by
GlaxoSmithKline · Sirtris, a GSK Company

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT01453491 Feb 2012 → Mar 2013 ulcerative colitis Sirtris, a GSK Company Completed No outcome recorded
Phase 1 NCT01031108 May 2010 → Oct 2011 type 2 diabetes mellitus Sirtris, a GSK Company Completed No outcome recorded
Phase 1 NCT00920660 Apr → Jun 2009 chronic obstructive pulmonary disease GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT00938275 Jan → Mar 2009 type 2 diabetes mellitus Sirtris, a GSK Company Completed No outcome recorded
Phase 1 NCT00937872 Nov → Dec 2008 type 2 diabetes mellitus Sirtris, a GSK Company Completed No outcome recorded
Phase 1 NCT00933530 May → Nov 2008 type 2 diabetes mellitus Sirtris, a GSK Company Completed No outcome recorded
Also used as a comparator or background therapy in 8 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT01702493 Comparator Oct → Dec 2012 psoriasis Sirtris, a GSK Company Completed No outcome recorded
Phase 1 NCT01039909 Comparator Jan → Feb 2011 muscular atrophy GlaxoSmithKline Withdrawn No outcome recorded
Phase 1 NCT01014117 Comparator Dec 2009 → May 2010 infectious disease with sepsis GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT00964340 Comparator Oct 2009 → Apr 2010 muscular atrophy GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT00933062 Comparator Mar → May 2009 type 2 diabetes mellitus GlaxoSmithKline Completed No outcome recorded
Phase 23 trials
Phase 2 NCT01154101 Comparator Jun 2010 → Nov 2011 psoriasis Sirtris, a GSK Company Completed No outcome recorded
Phase 2 NCT01018017 Comparator Mar → Dec 2010 type 2 diabetes mellitus GlaxoSmithKline Completed No outcome recorded
Phase 2 NCT00937326 Comparator Aug 2009 → Sep 2010 type 2 diabetes mellitus Sirtris, a GSK Company Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 14 sources stand behind the page.

FieldValueCited text
Known as SRT2104 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00938275
13

NCT00933062

NCT01453491

NCT00920660

NCT01031108

NCT01039909

NCT01018017

NCT00933530

NCT01154101

NCT00937326

NCT00964340

NCT01014117

NCT00937872

NCT01702493

Action Activate “SRT2104 is a potent small molecule activator of SIRT1” NCT01014117
Modality Small molecule “SRT2104 is a potent small molecule activator of SIRT1” NCT01014117
Route Oral “single, oral doses of SRT2104 (250 mg, 500 mg, 1000 mg, 2000 mg)” NCT00920660
Target SIRT1 “SRT2104 is a potent small molecule activator of SIRT1NCT01014117