Drugs / Piclidenoson
last change Jun 2026 re-read 2 minutes ago

Piclidenoson

also known as CF101 · ALB-7208 · IB-MECA

Small molecule targets ADORA3 via activation

Developed for
psoriasis · rheumatoid arthritis · dry eye syndrome · COVID-19 · glaucoma · intermediate uveitis · ocular hypertension · oculocerebrorenal syndrome
+2 more · osteoarthritis, knee · posterior uveitis
Investigated by
Can-Fite BioPharma · Rabin Medical Center

Trials 15 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 210 trials
Phase 2 NCT07410455 Jun 2026 → Aug 2027 expected oculocerebrorenal syndrome Can-Fite BioPharma Not yet recruiting No outcome recorded
Phase 2 NCT04333472 Jan 2021 → Mar 2022 COVID-19 Can-Fite BioPharma Completed No outcome recorded
Phase 2 NCT01905124 Jan → Sep 2019 intermediate uveitis, posterior uveitis Can-Fite BioPharma Withdrawn No outcome recorded
Phase 2 NCT00837291 Nov → Dec 2018 osteoarthritis, knee Can-Fite BioPharma Withdrawn No outcome recorded
Phase 2 NCT01034306 Oct 2010 → Dec 2013 rheumatoid arthritis Can-Fite BioPharma Completed No outcome recorded
Phase 2 NCT01033422 Oct 2010 → Dec 2016 glaucoma, ocular hypertension Can-Fite BioPharma Completed No outcome recorded
Phase 2 NCT00556894 Feb 2008 → Mar 2009 rheumatoid arthritis Can-Fite BioPharma Completed No outcome recorded
Phase 2 NCT00428974 Jun 2007 → Sep 2009 psoriasis Can-Fite BioPharma Completed No outcome recorded
Phase 2 NCT00349466 Jan 2007 → May 2009 dry eye syndrome Can-Fite BioPharma Completed No outcome recorded
Phase 2 NCT00280917 Jun 2006 → Apr 2007 rheumatoid arthritis Can-Fite BioPharma Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT01265667 Jul 2011 → Mar 2015 psoriasis Can-Fite BioPharma Completed No outcome recorded
Phase 34 trials
Phase 3 NCT06643260 Jun 2025 → Dec 2027 expected psoriasis Can-Fite BioPharma Not yet recruiting No outcome recorded
Phase 3 NCT03168256 Sep 2018 → Jan 2022 psoriasis Can-Fite BioPharma Completed No outcome recorded
Phase 3 NCT02647762 Oct 2017 → Nov 2020 rheumatoid arthritis Can-Fite BioPharma Terminated No outcome recorded
Phase 3 NCT01235234 Jul 2011 → Nov 2013 dry eye syndrome Can-Fite BioPharma Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 17 sources stand behind the page.

FieldValueCited text
Known as Piclidenoson “We investigated the efficacy/safety of piclidenoson (CF101), an orally bioavailable A3AR agonist that inhibits IL-17 and IL-23 production in keratinocytes, in...” PMID 38279575 Jan 2024
3

NCT07410455

NCT04333472

NCT06643260

Known as ALB-7208 ChEMBL registry synonym — accepted as the source's own label CHEMBL3989873
Known as CF101 “We investigated the efficacy/safety of piclidenoson (CF101), an orally bioavailable A3AR agonist that inhibits IL-17 and IL-23 production in keratinocytes, in...” PMID 38279575 Jan 2024
13

“A Phase 3, Randomized, Double-Blind, Placebo-Controlled Study of the Efficacy and Safety of Daily Piclidenoson (CF101) Administered Orally in Subjects With Moderate-to-Severe...” NCT06643260

“Piclidenoson (CF101) open-label treated patients” NCT07410455

NCT02647762

NCT01265667

NCT00280917

NCT00556894

NCT01235234

NCT00428974

NCT00349466

NCT01034306

NCT01033422

NCT00837291

NCT01905124

Known as IB-MECA ChEMBL registry synonym — accepted as the source's own label CHEMBL3989873
Action Activate “A(3) adenosine receptor agonist” PMID 20304499 Mar 2010
1

“Adenosine A3 receptor agonist” CHEMBL3989873

Modality Small molecule CHEMBL3989873
Route Oral “CF101 0.1 mg, CF101 1 mg, CF101 4 mg, or placebo given orally q12h for 12 weeks” NCT00280917
Target ADORA3 “Adenosine A3 receptor agonist” CHEMBL3989873