Drugs / Tozadenant
last change Jan 2018 re-read 2 minutes ago

Tozadenant

Small molecule targets ADORA2A via inhibition

Developed for
Parkinson disease · cocaine dependence
Investigated by
Biotie Therapies Inc. · Acorda Therapeutics · PRA Health Sciences · Tandem Labs · Xceleron Inc

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT03200080 Sep → Nov 2017 substance abuse Biotie Therapies Inc. Terminated No outcome recorded
Phase 1 NCT03212313 Jun → Dec 2017 Biotie Therapies Inc. Terminated No outcome recorded
Phase 1 NCT02240290 Sep → Oct 2013 Biotie Therapies Inc. Completed No outcome recorded
Phase 21 trial
Phase 2 NCT00605553 Apr 2008 → May 2009 Parkinson disease Biotie Therapies Inc. Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT01283594 Mar 2011 → Oct 2012 Parkinson disease Biotie Therapies Inc. Completed No outcome recorded
Phase 32 trials
Phase 3 NCT03051607 Apr 2017 → Jan 2018 Parkinson disease Biotie Therapies Inc. Terminated No outcome recorded
Phase 3 NCT02453386 Jul 2015 → Jan 2018 Parkinson disease Biotie Therapies Inc. Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 0 NCT00783276 Comparator Oct 2008 → Jan 2013 cocaine dependence Virginia Commonwealth University Completed No outcome recorded

Evidence & citations 10 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as Tozadenant ClinicalTrials.gov intervention name — accepted as the source's own label NCT03212313
6

NCT02453386

NCT01283594

NCT00605553

NCT02240290

NCT03051607

NCT03200080

Known as A-2A (3) ChEMBL registry synonym — accepted as the source's own label CHEMBL2105747
Known as RO-4494351 ChEMBL registry synonym — accepted as the source's own label CHEMBL2105747
Known as RO-4494351-000 ChEMBL registry synonym — accepted as the source's own label CHEMBL2105747
Known as RO-4494351-002 ChEMBL registry synonym — accepted as the source's own label CHEMBL2105747
Known as SYN115 “Tozadenant (SYN115) is an oral, selective adenosine A2A receptor antagonist that improves motor function in animal models of Parkinson's disease.” PMID 25008546 Jul 2014
1

NCT00783276

Action Inhibit “Adenosine A2a receptor antagonist” CHEMBL2105747
1

“adenosine A(2a) antagonist” PMID 21123574 Dec 2010

Modality Small molecule CHEMBL2105747
Route Oral “Tozadenant 20 mg oral capsules” NCT00605553
Target ADORA2A “Adenosine A2a receptor antagonist” CHEMBL2105747