Drugs / Sevabertinib
last change Mar 2026 re-read 2 minutes ago

Sevabertinib

also known as BAY 2927088

Small molecule targets EGFR

Developed for
non-small cell lung carcinoma · cancer · lung cancer
Investigated by
Bayer

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) HYRNUO 2025-11-19 fda.gov

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT07102095 Jul → Dec 2025 liver disorder Bayer Completed No outcome recorded
Phase 1 NCT06360211 Apr → Jun 2024 non-small cell lung carcinoma Bayer Completed No outcome recorded
Phase 1 NCT06348888 Apr → Jun 2024 non-small cell lung carcinoma Bayer Completed No outcome recorded
Phase 1 NCT06378658 Mar → Jun 2024 non-small cell lung carcinoma Bayer Completed No outcome recorded
Phase 1 NCT06329895 Mar → Jun 2024 non-small cell lung carcinoma Bayer Completed No outcome recorded
Phase 1 NCT06221475 Jan → Apr 2024 non-small cell lung carcinoma Bayer Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT05099172 Oct 2021 → Mar 2026 overdue non-small cell lung carcinoma Bayer Recruiting No outcome recorded
Phase 21 trial
Phase 2 NCT06760819 Feb 2025 → Feb 2027 expected cancer Bayer Recruiting No outcome recorded
Phase 31 trial
Phase 3 NCT06452277 Aug 2024 → Oct 2027 expected lung cancer Bayer Recruiting No outcome recorded
Phase not stated1 trial
NCT06761976 non-small cell lung carcinoma Bayer Available No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as Sevabertinib Sevabertinib is an oral, reversible tyrosine kinase inhibitor that has shown anti-HER2 activity in preclinical models.” PMID 41104928 Oct 2025
3

NCT06761976

NCT06452277

NCT07102095

Known as BAY 2927088 “A Phase 1 Open Label, Two-arm, Fixed Sequence, Crossover Study to Investigate the Effects of Itraconazole and Carbamazepine on the Pharmacokinetics of BAY 2927088 in Healthy...” NCT06348888
9

“A Phase 1, Open Label, Fixed Sequence, Crossover Study to Investigate the Effect of BAY 2927088 on the Pharmacokinetics of Midazolam in Healthy Participants” NCT06360211

“A Phase 1, Open-label, Single-dose Study to Assess the Influence of Hepatic Impairment on the Pharmacokinetics of of Sevabertinib (BAY 2927088)” NCT07102095

“The study treatment, sevabertinib (BAY2927088), is expected to block the mutated EGFR and HER2 proteins which may stop the spread of NSCLC.” NCT05099172

NCT06221475

NCT06329895

NCT06378658

NCT06348888

NCT06360211

NCT06760819

Action Inhibit “The study treatment, sevabertinib (BAY2927088), is expected to block the mutated EGFR and HER2 proteins which may stop the spread of NSCLC.” NCT05099172
Modality Small molecule “Sevabertinib is an oral, reversible tyrosine kinase inhibitor that has shown anti-HER2 activity in preclinical models.” PMID 41104928 Oct 2025
1

CHEMBL6068074

Route Oral “The participants in this study will take the study treatment BAY2927088 in 3-week periods called "cycles". They will in general take BAY2927088 once or twice daily as a...” NCT05099172
Target EGFR “The study treatment, sevabertinib (BAY2927088), is expected to block the mutated EGFR and HER2 proteins which may stop the spread of NSCLC.” NCT05099172