Drugs / Darovasertib
last change Jan 2026 re-read 2 minutes ago

Darovasertib

also known as IDE196 · LXS196 · NVP-LXS-196

Small molecule

Developed for
uveal melanoma · colorectal cancer · cutaneous melanoma · ocular melanoma
Investigated by
IDEAYA Biosciences · Novartis Pharmaceuticals · St Vincent's Hospital, Sydney

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT02601378 Feb 2016 → Jan 2022 uveal melanoma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT03947385 Jun 2019 → Jan 2027 expected colorectal cancer, cutaneous melanoma, uveal melanoma IDEAYA Biosciences Recruiting No outcome recorded
Phase 22 trials
Phase 2 NCT05907954 Jul 2023 → Apr 2027 expected uveal melanoma IDEAYA Biosciences Active not recruiting No outcome recorded
Phase 2 NCT05187884 May 2022 → Jan 2025 ocular melanoma St Vincent's Hospital, Sydney Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT05987332 Oct 2023 → Jan 2027 expected uveal melanoma IDEAYA Biosciences Active not recruiting No outcome recorded
Phase 31 trial
Phase 3 NCT07015190 Jan 2026 → Oct 2030 expected uveal melanoma IDEAYA Biosciences Recruiting No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as Darovasertib “IDE196 (Darovasertib) in Combination With Crizotinib as First-line Therapy in Metastatic Uveal Melanoma” NCT05987332
3

NCT05187884

NCT05907954

NCT07015190

Known as IDE196 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03947385
1

NCT05987332

Known as LXS196 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02601378
Known as NVP-LXS-196 ChEMBL registry synonym — accepted as the source's own label CHEMBL3982723
Action Inhibit “Protein Kinase C Inhibitor” NCT02601378
Modality Small molecule CHEMBL3982723
Route Oral “LXS196, an Oral Protein Kinase C Inhibitor” NCT02601378