Drugs / RUPITASERTIB
last change Aug 2018 re-read 2 minutes ago

RUPITASERTIB

also known as M-2698 · MSC2363318A

Small molecule targets AKT1, AKT3 via inhibition

Developed for
cancer
Investigated by
EMD Serono

Trials 1 · a red edge is where a trial was stopped

20142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT01971515 Dec 2013 → Aug 2018 cancer EMD Serono Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 2 sources stand behind the page.

FieldValueCited text
Known as RUPITASERTIB ChEMBL registry synonym — accepted as the source's own label CHEMBL4871106
Known as M-2698 ChEMBL registry synonym — accepted as the source's own label CHEMBL4871106
Known as MSC2363318A ClinicalTrials.gov intervention name — accepted as the source's own label NCT01971515
Action Inhibit “Serine/threonine-protein kinase AKT3 inhibitor” CHEMBL4871106
1

“Serine/threonine-protein kinase AKT inhibitor” CHEMBL4871106

Modality Small molecule CHEMBL4871106
Route Oral “MSC2363318A will be administered orally once daily” NCT01971515
Target AKT1 “Serine/threonine-protein kinase AKT inhibitor” CHEMBL4871106
Target AKT3 “Serine/threonine-protein kinase AKT3 inhibitor” CHEMBL4871106