Drugs / OP-3136
last change Dec 2024 re-read 2 minutes ago

OP-3136

targets KAT6A, KAT6B via inhibition

Developed for
castration-resistant prostate carcinoma · estrogen-receptor positive breast cancer · non-small cell lung carcinoma
Investigated by
Olema Pharmaceuticals, Inc.

Trials 1 · a red edge is where a trial was stopped

202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT06784193 Dec 2024 → May 2027 expected castration-resistant prostate carcinoma, estrogen-receptor positive breast cancer, non-small cell lung carcinoma, progesterone-receptor positive breast cancer Olema Pharmaceuticals, Inc. Recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 1 source stands behind the page.

FieldValueCited text
Known as OP-3136 ClinicalTrials.gov intervention name — accepted as the source's own label NCT06784193
Action Inhibit “Selective inhibitor of HAT enzymes KAT6A and KAT6B” NCT06784193
Route Oral “administered orally once daily” NCT06784193
Target KAT6A “Selective inhibitor of HAT enzymes KAT6A and KAT6B” NCT06784193
Target KAT6B “Selective inhibitor of HAT enzymes KAT6A and KAT6BNCT06784193