Drugs / APLAVIROC
last change Oct 2007 re-read 2 minutes ago

APLAVIROC

Small molecule targets CCR5 via inhibition

Developed for
HIV infectious disease
Investigated by
GlaxoSmithKline · ViiV Healthcare · National Institute of Allergy and Infectious Diseases (NIAID)

Trials 6 · a red edge is where a trial was stopped

200420052006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 23 trials
Phase 2 NCT00104429 Jan 2005 → Jan 2006 HIV infectious disease ViiV Healthcare Terminated No outcome recorded
Phase 2 NCT00102778 Dec 2004 → Sep 2007 HIV infectious disease ViiV Healthcare Terminated No outcome recorded
Phase 2 NCT00076284 Jan 2004 → Mar 2005 HIV infectious disease National Institute of Allergy and Infectious Diseases (NIAID) Completed No outcome recorded
Phase 33 trials
Phase 3 NCT00197145 Jul 2005 → Sep 2007 HIV infectious disease ViiV Healthcare Terminated No outcome recorded
Phase 3 NCT00297076 Jul 2005 → Oct 2007 HIV infectious disease GlaxoSmithKline Terminated No outcome recorded
Phase 3 NCT00197197 Jul → Oct 2005 HIV infectious disease GlaxoSmithKline Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 3 NCT00123890 Background Jun → Oct 2005 HIV infectious disease GlaxoSmithKline Terminated No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as APLAVIROC ChEMBL registry synonym — accepted as the source's own label CHEMBL1255794
Known as AK-602 ChEMBL registry synonym — accepted as the source's own label CHEMBL1255794
Known as Aplaviroc hcl ChEMBL registry synonym — accepted as the source's own label CHEMBL1255794
Known as APLAVIROC HYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL1255794
Known as GSK-873140 ChEMBL registry synonym — accepted as the source's own label CHEMBL1255794
Known as GW-873140A ChEMBL registry synonym — accepted as the source's own label CHEMBL1255794
Known as GW873140 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00197197
6

NCT00123890

NCT00297076

NCT00197145

NCT00102778

NCT00104429

NCT00076284

Action Inhibit “GW873140 is intended to block the CCR5 receptor so that HIV-1 cannot enter the cell.” NCT00076284
Modality Small molecule CHEMBL1255794
Route Oral “following oral dosing” NCT00076284
Target CCR5 “block the CCR5 receptor” NCT00076284