Drugs / LNS8801
last change 20 days ago re-read 2 minutes ago

LNS8801

also known as CHEMBL569766 · ML051

Small molecule targets GPER1 via activation

Developed for
cancer · cutaneous melanoma
Investigated by
Linnaeus Therapeutics, Inc. · Merck Sharp & Dohme LLC

Trials 2 · a red edge is where a trial was stopped

2020202120222023202420252026202720282029
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/21 trial
Phase 1/2 NCT04130516 Oct 2019 → Jun 2026 overdue cancer Linnaeus Therapeutics, Inc. Active not recruiting No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT06624644 Aug 2025 → Feb 2029 expected cutaneous melanoma Linnaeus Therapeutics, Inc. Recruiting No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 3 sources stand behind the page.

FieldValueCited text
Known as LNS8801 ClinicalTrials.gov intervention name — accepted as the source's own label NCT06624644
1

NCT04130516

Known as CHEMBL569766 ChEMBL registry synonym — accepted as the source's own label CHEMBL569766
Known as ML051 ChEMBL registry synonym — accepted as the source's own label CHEMBL569766
Action Activate “selective agonist of GPER” NCT04130516
Modality Small molecule CHEMBL569766
Route Oral “LNS8801 will be administered orally” NCT04130516
Target GPER “selective agonist of GPERNCT04130516