Drugs / NIR178

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT04237649 Feb 2020 → Sep 2023 cancer Novartis Pharmaceuticals Terminated No outcome recorded
Phase 14 trials
Phase 1 NCT04895748 Nov 2021 → Feb 2026 clear cell renal carcinoma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1 NCT03742349 Jan 2019 → Feb 2023 triple-negative breast carcinoma Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1 NCT03549000 Jul 2018 → Oct 2022 colorectal cancer, non-small cell lung carcinoma, ovarian cancer, pancreatic ductal adenocarcinoma +3 Novartis Pharmaceuticals Terminated No outcome recorded
Phase 1 NCT02403193 Oct 2015 → Oct 2021 non-small cell lung carcinoma Palobiofarma SL Completed No outcome recorded
Phase 21 trial
Phase 2 NCT03207867 Aug 2017 → Feb 2023 colorectal cancer, diffuse large B-cell lymphoma, head and neck cancer, malignant pancreatic neoplasm +6 Novartis Pharmaceuticals Terminated No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as NIR178 “Phase I Study of Taminadenant (PBF509/NIR178), an Adenosine 2A Receptor Antagonist, with or without Spartalizumab (PDR001), in Patients with Advanced Non-Small Cell Lung Cancer.” PMID 35254415 Jun 2022
5

NCT04237649

NCT03549000

NCT03742349

NCT03207867

NCT04895748

Known as PBF509 “Phase I Study of Taminadenant (PBF509/NIR178), an Adenosine 2A Receptor Antagonist, with or without Spartalizumab (PDR001), in Patients with Advanced Non-Small Cell Lung Cancer.” PMID 35254415 Jun 2022
Known as Taminadenant “Phase I Study of Taminadenant (PBF509/NIR178), an Adenosine 2A Receptor Antagonist, with or without Spartalizumab (PDR001), in Patients with Advanced Non-Small Cell Lung Cancer.” PMID 35254415 Jun 2022
Action Inhibit “Taminadenant (PBF509/NIR178) is an A2AR antagonist able to reactivate the antitumor immune response.” PMID 35254415 Jun 2022
Route Oral “NIR178 was administered orally twice daily (BID) as a capsule” NCT03207867