Drugs / Rovadicitinib
last change Apr 2026 re-read 2 minutes ago

Rovadicitinib

also known as TQ05105

Small molecule targets ROCK2 via inhibition

Developed for
chronic graft versus host disease · myelofibrosis
Investigated by
Chia Tai Tianqing Pharmaceutical Group Co., Ltd.

Trials 4 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT06388759 Aug 2022 → Aug 2025 myelofibrosis Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Terminated No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT04944043 Jun 2021 → Jun 2023 overdue chronic graft versus host disease Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Active not recruiting No outcome recorded
Phase 21 trial
Phase 2 NCT06300320 May 2024 → Oct 2025 overdue chronic graft versus host disease Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Recruiting No outcome recorded
Phase 31 trial
Phase 3 NCT06682169 Nov 2024 → Oct 2029 expected chronic graft versus host disease Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Recruiting No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as Rovadicitinib Rovadicitinib (TQ05105) is a novel, oral dual Janus kinase 1/2 and rho-associated coiled-coil-containing protein kinase-1/2 inhibitor targeting inflammatory and fibrotic...” PMID 40009501 Jun 2025
3

Rovadicitinib (TQ05105) is a novel, oral dual JAK 1/2 and Rho-associated kinases (ROCK) 1/2 inhibitor targeting inflammatory and fibrotic components of cGVHD.” NCT06300320

Rovadicitinib (TQ05105) is a first-in-class, oral, small-molecule Janus kinase (JAK)/Rho-associated kinase (ROCK) inhibitor.” PMID 40752760 Aug 2025

NCT06682169

Known as TQ05105 “Rovadicitinib (TQ05105) is a novel, oral dual Janus kinase 1/2 and rho-associated coiled-coil-containing protein kinase-1/2 inhibitor targeting inflammatory and fibrotic...” PMID 40009501 Jun 2025
2

“Rovadicitinib (TQ05105) is a novel, oral dual JAK 1/2 and Rho-associated kinases (ROCK) 1/2 inhibitor targeting inflammatory and fibrotic components of cGVHD.” NCT06300320

“Rovadicitinib (TQ05105) is a first-in-class, oral, small-molecule Janus kinase (JAK)/Rho-associated kinase (ROCK) inhibitor.” PMID 40752760 Aug 2025

Action Inhibit “TQ05105 tablet is a Janus Kinase (JAK) inhibitor, which can inhibit the abnormal activation of JAK 2-V617F mutation, thereby inhibiting the sustained abnormal activation of JAK...” NCT04944043
Modality Small molecule “Rovadicitinib (TQ05105) is a first-in-class, oral, small-molecule Janus kinase (JAK)/Rho-associated kinase (ROCK) inhibitor.” PMID 40752760 Aug 2025
Route Oral “TQ05105 tablet 10mg given orally” NCT04944043
Target ROCK2 “It can inhibit the sustained abnormal activation of the Janus kinase (JAK) signal transducer and activator of transcription (JAK-STAT) pathway and also inhibit Rho associated...” NCT06682169