Drugs / Rostafuroxin
last change Feb 2018 re-read 2 minutes ago

Rostafuroxin

also known as Rostafuroxina · Rostafuroxine

Small molecule

Developed for
essential hypertension
Investigated by
RostaQuo S.p.A. · Windtree Therapeutics · sigma-tau i.f.r. S.p.A.

Trials 3 · a red edge is where a trial was stopped

20052006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT03217825 Dec 2015 → Feb 2018 essential hypertension Windtree Therapeutics Completed No outcome recorded
Phase 2 NCT01320397 May 2011 → Jul 2012 essential hypertension RostaQuo S.p.A. Unknown No outcome recorded
Phase 2 NCT00415038 Feb 2005 → Apr 2007 essential hypertension sigma-tau i.f.r. S.p.A. Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as Rostafuroxin ClinicalTrials.gov intervention name — accepted as the source's own label NCT01320397
2

NCT03217825

NCT00415038

Known as Rostafuroxina ChEMBL registry synonym — accepted as the source's own label CHEMBL2068971
Known as Rostafuroxine ChEMBL registry synonym — accepted as the source's own label CHEMBL2068971
Action Inhibit “which selectively antagonizes the effects of endogenous ouabain (EO) on Na+,K+-ATPase and mutated adducin” PMID 21235787 Jan 2011
Modality Small molecule “rostafuroxin, a digitoxygenin derivative” PMID 21235787 Jan 2011
Route Oral “The antihypertensive effect of rostafuroxin is long-lasting since it is still present 24 hours after oral administration” NCT01320397