Drugs / istiratumab
last change Jan 2020 re-read 2 minutes ago

istiratumab

also known as MM-141 · MM-005

Monoclonal antibody targets ERBB3, IGF1R via inhibition

Developed for
colorectal cancer · head and neck squamous cell carcinoma · hepatocellular carcinoma · malignant pancreatic neoplasm · non-small cell lung carcinoma
Investigated by
Merrimack Pharmaceuticals

Trials 3 · a red edge is where a trial was stopped

201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT02538627 Aug 2015 → Oct 2016 colorectal cancer, head and neck squamous cell carcinoma, non-small cell lung carcinoma Merrimack Pharmaceuticals Terminated No outcome recorded
Phase 1 NCT01733004 Nov 2012 → Jan 2016 hepatocellular carcinoma Merrimack Pharmaceuticals Completed No outcome recorded
Phase 21 trial
Phase 2 NCT02399137 May 2015 → Aug 2018 malignant pancreatic neoplasm Merrimack Pharmaceuticals Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as istiratumab “Randomized, double-blind, placebo-controlled phase II study of istiratumab (MM-141) plus nab-paclitaxel and gemcitabine versus nab-paclitaxel and gemcitabine in front-line...” PMID 31912800 Jan 2020
Known as MM-005 ChEMBL registry synonym — accepted as the source's own label CHEMBL3989990
Known as MM-141 “Randomized, double-blind, placebo-controlled phase II study of istiratumab (MM-141) plus nab-paclitaxel and gemcitabine versus nab-paclitaxel and gemcitabine in front-line...” PMID 31912800 Jan 2020
2

NCT01733004

NCT02538627

Action Inhibit “dual blockade of the insulin-like growth factor-1 receptor (IGF-1R) and HER3 pathways” PMID 31912800 Jan 2020
1

“Receptor tyrosine-protein kinase erbB-3 inhibitor” CHEMBL3989990

Modality Monoclonal antibody “istiratumab, an IGF-1R- and ErbB3-bispecific antibody” PMID 31912800 Jan 2020
1

CHEMBL3989990

Route Intravenous “2.8 g intravenously (i.v.) every 2 weeks” PMID 31912800 Jan 2020
Target ERBB3 “Receptor tyrosine-protein kinase erbB-3 inhibitor” CHEMBL3989990
Target IGF1R “dual blockade of the insulin-like growth factor-1 receptor (IGF-1R) and HER3 pathways” PMID 31912800 Jan 2020