Drugs / CARBAMOYLCHOLINE
last change Dec 2025 re-read 2 minutes ago

CARBAMOYLCHOLINE

Small molecule targets CHRM3 via activation

Developed for
presbyopia
Investigated by
Danish Headache Center · Zhaoke (Guangzhou) Ophthalmology Pharmaceutical Ltd.

Regulatory milestones approvals, filings & regulatory actions · 2 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansion US (FDA) MIOSTAT 1995-08-18 fda.gov
Approved US (FDA) MIOSTAT 1972-09-28 fda.gov

Trials 2 · a red edge is where a trial was stopped

197219731974197519761977197819791980198119821983198419851986198719881989199019911992199319941995199619971998199920002001200220032004200520062007200820092010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 21 trial
Phase 2 NCT06948357 Mar → Sep 2025 overdue presbyopia Zhaoke (Guangzhou) Ophthalmology Pharmaceutical Ltd. Recruiting No outcome recorded
Phase not applicable1 trial
NCT00564408 Aug 2007 → Oct 2008 headache disorder Danish Headache Center Completed No outcome recorded
Also used as a comparator or background therapy in 4 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 21 trial
Phase 2 NCT04774237 Comparator Mar → Oct 2021 presbyopia Visus Therapeutics Completed No outcome recorded
Phase 32 trials
Phase 3 NCT05270863 Comparator Mar 2022 → Mar 2023 presbyopia Visus Therapeutics Completed No outcome recorded
Phase 3 NCT05135286 Comparator Mar 2022 → Mar 2025 presbyopia Visus Therapeutics Completed No outcome recorded
Phase not applicable1 trial
NCT04274413 Background Feb 2021 CFTR-related disorder, cystic fibrosis The Hospital for Sick Children Withdrawn No outcome recorded

Evidence & citations 13 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as CARBAMOYLCHOLINE ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Known as Carbachol “Under the second probe, first injection carbachol will be given in one small area of the skin.” NCT04274413
5

NCT04774237

NCT00564408

NCT05135286

NCT06948357

NCT05270863

Known as Carbachol chloride ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Known as CARBACHOL PF “BRIMOCHOL PF eye drops, CARBACHOL PF eye drops, Brimonidine eye drops and Placebo were administered in 7 treatment sequences in various combinations and doses” NCT06948357
Known as Carbacol ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Known as Carbastat ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Known as Doryl ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Known as Miostat ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Known as NSC-32865 ChEMBL registry synonym — accepted as the source's own label CHEMBL965
Action Activate “Muscarinic acetylcholine receptor M3 agonist” CHEMBL965
Modality Small molecule CHEMBL965
Route Intravenous “infused intravenously” NCT00564408
Target CHRM3 “Muscarinic acetylcholine receptor M3 agonist” CHEMBL965