Drugs / Firsocostat
last change Dec 2024 re-read 2 minutes ago

Firsocostat

also known as FIR · GS-0976 · GS-ACC · ND-630 · Ndi-010976

Small molecule

Developed for
metabolic dysfunction-associated steatohepatitis · NAFLD1
Investigated by
Gilead Sciences · Novo Nordisk A/S · Nimbus Apollo

Trials 7 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT02891408 Sep 2016 → May 2019 metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded
Phase 1 NCT02876796 Aug → Sep 2015 Gilead Sciences Completed No outcome recorded
Phase 25 trials
Phase 2 NCT04971785 Aug 2021 → Nov 2024 metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded
Phase 2 NCT03987074 Jul 2019 → Jul 2020 metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded
Phase 2 NCT03449446 Mar 2018 → Oct 2019 metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded
Phase 2 NCT02856555 Aug 2016 → Jul 2017 metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded
Phase 2 NCT02781584 Jun 2016 → Dec 2020 NAFLD1, metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded

Press releases naming this drug 2 releases

DateIssuerRelease
2017-10-24 Gilead Sciences Gilead Announces Phase 2 Results for GS-0976 in Nonalcoholic Steatohepatitis (NASH) gilead.com
2017-04-21 Gilead Sciences Gilead Presents Proof-of-Concept Data for GS-0976 in Nonalcoholic Steatohepatitis (NASH) at The International Liver Congress™ 2017 gilead.com

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as Firsocostat “the acetyl-CoA carboxylase inhibitor firsocostat (FIR) improved liver histology and biomarkers in NASH with advanced fibrosis” PMID 34999207 Jan 2022
5

Firsocostat (FIR)” NCT03449446

NCT02856555

NCT03987074

NCT04971785

NCT02891408

Known as FIR “the acetyl-CoA carboxylase inhibitor firsocostat (FIR) improved liver histology and biomarkers in NASH with advanced fibrosis” PMID 34999207 Jan 2022
2

“Cilofexor (CILO)/Firsocostat (FIR)” NCT04971785

Firsocostat (FIR)” NCT03449446

Known as GS-0976 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02876796
Known as GS-ACC ChEMBL registry synonym — accepted as the source's own label CHEMBL3407547
Known as ND-630 ChEMBL registry synonym — accepted as the source's own label CHEMBL3407547
Known as Ndi-010976 ChEMBL registry synonym — accepted as the source's own label CHEMBL3407547
Action Inhibit “the acetyl-CoA carboxylase inhibitor firsocostat (FIR)” PMID 34999207 Jan 2022
Modality Small molecule CHEMBL3407547
Route Oral “Administered orally once daily” NCT02781584