Drugs / AZD5672
last change Nov 2010 re-read 2 minutes ago

AZD5672

Small molecule targets CCR5 via inhibition

Developed for
rheumatoid arthritis
Investigated by
AstraZeneca · Quintiles, Inc.

Trials 8 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT00887770 Apr → Jul 2009 rheumatoid arthritis AstraZeneca Completed No outcome recorded
Phase 1 NCT00871767 Mar → May 2009 rheumatoid arthritis AstraZeneca Completed No outcome recorded
Phase 1 NCT00746837 Aug 2008 → Jan 2009 AstraZeneca Completed No outcome recorded
Phase 1 NCT00723424 Jul → Dec 2008 AstraZeneca Completed No outcome recorded
Phase 1 NCT00722956 Jul → Aug 2008 AstraZeneca Completed No outcome recorded
Phase 1 NCT00715702 Jul 2008 → Feb 2009 impaired renal function disease AstraZeneca Completed No outcome recorded
Phase 1 NCT00711074 Jun → Jul 2008 rheumatoid arthritis AstraZeneca Completed No outcome recorded
Phase 21 trial
Phase 2 NCT00713544 Jul 2008 → Apr 2009 rheumatoid arthritis AstraZeneca Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as AZD5672 “Single Oral Doses of AZD5672 (600 mg and 150 mg)” NCT00887770
7

NCT00723424

NCT00746837

NCT00715702

NCT00722956

NCT00713544

NCT00711074

NCT00871767

Action Inhibit “AZD5672 was a highly potent and selective antagonist of CCR5” PMID 20662070 Nov 2010
Modality Small molecule “a small-molecule antagonist of CCR5” PMID 20662070 Nov 2010
Route Oral “Treatment arms were AZD5672 (20, 50, 100, or 150 mg orally, once daily), matched placebo, or open-label etanercept (50 mg subcutaneously, once weekly).” PMID 20662070 Nov 2010
Target CCR5 “blocking the chemokine receptor CCR5PMID 20662070 Nov 2010