Drugs / ENVUCITINIB
last change Jul 2026 re-read 2 minutes ago

ENVUCITINIB

also known as ESK-001 · Envudeucitinib

Small molecule targets TYK2 via inhibition

Developed for
psoriasis · intermediate uveitis · panuveitis · posterior uveitis · systemic lupus erythematosus
Investigated by
Alumis Inc

Trials 12 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT06952634 Apr 2025 → Mar 2026 Alumis Inc Completed No outcome recorded
Phase 1 NCT06962774 Apr → Aug 2025 impaired renal function disease Alumis Inc Completed No outcome recorded
Phase 1 NCT07378579 Jun → Aug 2024 Alumis Inc Completed No outcome recorded
Phase 1 NCT05431634 May → Dec 2022 Alumis Inc Completed No outcome recorded
Phase 1 NCT05330858 Mar → Jun 2022 Alumis Inc Completed No outcome recorded
Phase 24 trials
Phase 2 NCT05966480 Jun 2023 → Jul 2026 overdue systemic lupus erythematosus Alumis Inc Active not recruiting No outcome recorded
Phase 2 NCT05953688 Jun 2023 → Aug 2024 intermediate uveitis, panuveitis, posterior uveitis Alumis Inc Terminated No outcome recorded
Phase 2 NCT05739435 Jan 2023 → Dec 2026 expected psoriasis Alumis Inc Active not recruiting No outcome recorded
Phase 2 NCT05600036 Sep 2022 → Jun 2023 psoriasis Alumis Inc Completed No outcome recorded
Phase 33 trials
Phase 3 NCT06846541 Jan 2025 → Nov 2028 expected psoriasis Alumis Inc Active not recruiting No outcome recorded
Phase 3 NCT06588738 Aug 2024 → Sep 2025 psoriasis Alumis Inc Completed No outcome recorded
Phase 3 NCT06586112 Jul 2024 → Sep 2025 psoriasis Alumis Inc Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 15 sources stand behind the page.

FieldValueCited text
Known as ENVUCITINIB ChEMBL registry synonym — accepted as the source's own label CHEMBL5499275
Known as Envudeucitinib ClinicalTrials.gov intervention name — accepted as the source's own label NCT06586112
5

NCT06952634

NCT05966480

NCT06846541

NCT06588738

NCT05739435

Known as ESK-001 “Patients will enter the long-term extension study following completion of one of the parent studies (ESK-001-016 or ESK-001-017) and will receive open-label ESK-001 twice daily...” NCT06846541
7

“Envudeucitinib (ESK-001), a highly selective, oral tyrosine kinase 2 inhibitor” PMID 41061968 Oct 2025

NCT05431634

NCT05600036

NCT05953688

NCT06962774

NCT05330858

NCT07378579

Action Inhibit “Highly selective, allosteric inhibition of TYK2 with oral ESK-001” PMID 40659116 Jul 2025
Modality Small molecule CHEMBL5499275
Route Oral “ESK-001 administered as an oral liquid” NCT05330858
Target TYK2 “Highly selective, allosteric inhibition of TYK2 with oral ESK-001” PMID 40659116 Jul 2025