Drugs / PADNARSERTIB
last change Oct 2025 re-read 2 minutes ago

PADNARSERTIB

also known as KPT-9274 · ATG-019 · Pak4-in-1

Small molecule targets NAMPT, PAK4

Developed for
non-Hodgkin lymphoma · cancer · acute myeloid leukemia
Investigated by
Antengene Therapeutics Limited · Karyopharm Therapeutics Inc

Trials 2 · a red edge is where a trial was stopped

2017201820192020202120222023202420252026
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT04281420 Apr 2020 → Oct 2023 non-Hodgkin lymphoma Antengene Therapeutics Limited Terminated No outcome recorded
Phase 1 NCT02702492 Jun 2016 → Jan 2021 cancer, non-Hodgkin lymphoma Karyopharm Therapeutics Inc Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT04914845 Comparator Aug 2021 → Jul 2025 acute myeloid leukemia University of Colorado, Denver Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as PADNARSERTIB ChEMBL registry synonym — accepted as the source's own label CHEMBL4297467
Known as ATG-019 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04281420
Known as KPT-9274 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04914845
1

NCT02702492

Known as Pak4-in-1 ChEMBL registry synonym — accepted as the source's own label CHEMBL4297467
Action Inhibit “dual inhibitor of PAK4 and NAMPT” NCT02702492
Modality Small molecule “KPT-9274 is a first-in-class orally bioavailable, non-competitive, small moleculeNCT04914845
Route Oral oral KPT-9274” NCT02702492
Target NAMPT “dual inhibitor of PAK4 and NAMPTNCT02702492
Target PAK4 “dual inhibitor of PAK4 and NAMPT” NCT02702492