Drugs / Edotecarin
last change Dec 2009 re-read 2 minutes ago

Edotecarin

Small molecule targets TOP1 via inhibition

Developed for
breast cancer · gastric cancer · esophageal cancer · glioblastoma · metastatic malignant neoplasm
Investigated by
Pfizer · Memorial Sloan Kettering Cancer Center · National Cancer Institute (NCI)

Trials 5 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT00072332 Aug 2003 → Dec 2005 esophageal cancer, gastric cancer Memorial Sloan Kettering Cancer Center Completed No outcome recorded
Phase 23 trials
Phase 2 NCT00087503 Apr 2004 → Jun 2005 gastric cancer Pfizer Completed No outcome recorded
Phase 2 NCT00067314 Jun 2003 → Jun 2007 breast cancer, metastatic malignant neoplasm Pfizer Completed No outcome recorded
Phase 2 NCT00070031 Jun 2003 → Apr 2006 breast cancer Memorial Sloan Kettering Cancer Center Completed No outcome recorded
Phase 31 trial
Phase 3 NCT00068952 Aug 2003 → Mar 2006 glioblastoma Pfizer Completed No outcome recorded

Evidence & citations 10 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as Edotecarin ClinicalTrials.gov intervention name — accepted as the source's own label NCT00087503
4

NCT00072332

NCT00068952

NCT00067314

NCT00070031

Known as Edotecarina ChEMBL registry synonym — accepted as the source's own label CHEMBL435191
Known as Edotecarine ChEMBL registry synonym — accepted as the source's own label CHEMBL435191
Known as J-107088 ChEMBL registry synonym — accepted as the source's own label CHEMBL435191
Known as PF-804950 ChEMBL registry synonym — accepted as the source's own label CHEMBL435191
Known as PHA-782615 “A Phase II Study Of Intravenous Edotecarin (PHA-782615) In Patients With Anthracycline- And Taxane Resistant Metastatic Breast Cancer” NCT00067314
1

“A Phase I Dose Escalation Study of Edotecarin (PHA-782615) and Cisplatin in Adult Patients With Advanced/Metastatic Solid Tumors” NCT00072332

Action Inhibit “DNA topoisomerase I inhibitor” CHEMBL435191
Modality Small molecule CHEMBL435191
Route Intravenous Intravenous Edotecarin” NCT00067314
Target TOP1 “DNA topoisomerase I inhibitor” CHEMBL435191