Drugs / ethacrynic acid
last change Jul 2017 re-read 2 minutes ago

ethacrynic acid

Small molecule targets SLC12A1 via inhibition

Developed for
glaucoma · urinary bladder cancer
Investigated by
Eugene Lee, MD · Molly Walsh · University of Kansas Medical Center

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) EDECRIN 1967-01-10 fda.gov

Trials 2 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT02852564 Aug 2016 → Jul 2017 urinary bladder cancer Eugene Lee, MD Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02051946 May 2014 → Oct 2015 glaucoma Molly Walsh Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 3 NCT01628731 Comparator Oct 2012 → Jul 2013 Bambino Gesù Hospital and Research Institute Completed No outcome recorded

Evidence & citations 14 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as Ethacrynic Acid ClinicalTrials.gov intervention name — accepted as the source's own label NCT02852564
2

NCT02051946

NCT01628731

Known as Acide etacrynique ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as Acido etacrinico ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as Edecrin ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as Etacrynic acid ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as Hydromedin ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as MK-595 ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as NSC-624008 ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as NSC-85791 ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Known as Reomax ChEMBL registry synonym — accepted as the source's own label CHEMBL456
Action Inhibit “Sodium-(potassium)-chloride cotransporter 2 inhibitor” CHEMBL456
Modality Small molecule CHEMBL456
Route Intravenous “ethacrynic acid, intravenous, continuous infusion, 0.2 mg/kg/h for 24 hours” NCT01628731
Target SLC12A1 “Sodium-(potassium)-chloride cotransporter 2 inhibitor” CHEMBL456