Drugs / ADOMEGLIVANT
last change Jul 2021 re-read 2 minutes ago

ADOMEGLIVANT

also known as LY2409021

Small molecule targets GCGR via inhibition

Developed for
type 2 diabetes mellitus · type 1 diabetes mellitus · post-surgical hypoinsulinemia
Investigated by
Eli Lilly and Company

Trials 15 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 111 trials
Phase 1 NCT02385084 Mar → May 2015 Eli Lilly and Company Terminated No outcome recorded
Phase 1 NCT02217618 Aug → Sep 2014 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01929109 Aug 2013 → Aug 2014 chronic renal failure syndrome Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01836198 May → Nov 2013 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01640834 Jul → Sep 2012 type 1 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01588366 Apr 2012 → Sep 2013 type 2 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01460368 Oct 2011 → Mar 2012 type 2 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01354496 Apr → Oct 2011 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01606397 Mar → Nov 2008 type 2 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01606423 Nov 2007 → Mar 2008 Eli Lilly and Company Completed No outcome recorded
Phase 24 trials
Phase 2 NCT02111096 Apr 2014 → Sep 2015 type 2 diabetes mellitus Eli Lilly and Company Terminated No outcome recorded
Phase 2 NCT02091362 Mar 2014 → Jan 2015 type 2 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT01241448 Jan 2011 → Feb 2012 type 2 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT00871572 Mar 2009 → Feb 2010 type 2 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
NCT02944110 Comparator Apr 2016 → Nov 2019 post-surgical hypoinsulinemia University Hospital, Gentofte, Copenhagen Unknown No outcome recorded
NCT02669524 Comparator Oct 2015 → Aug 2016 type 2 diabetes mellitus University Hospital, Gentofte, Copenhagen Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 19 sources stand behind the page.

FieldValueCited text
Known as ADOMEGLIVANT ChEMBL registry synonym — accepted as the source's own label CHEMBL3707351
Known as LY2409021 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01929109
16

NCT02111096

NCT01606397

NCT02669524

NCT02944110

NCT01354496

NCT01640834

NCT01606423

NCT00871572

NCT01588366

NCT02217618

NCT02091362

NCT02385084

NCT01606371

NCT01836198

NCT01460368

NCT01241448

Action Inhibit “glucagon receptor antagonist” PMID 26681715 Dec 2015
1

“Glucagon receptor antagonist” CHEMBL3707351

Modality Small molecule “a potent, selective small-molecule glucagon receptor antagonist” PMID 26681715 Dec 2015
Route Oral “once-daily oral administration of LY2409021” PMID 26681715 Dec 2015
Target GCGR “Glucagon receptor antagonist” CHEMBL3707351