Drugs / Brequinar
last change Jun 2022 re-read 2 minutes ago

Brequinar

Small molecule targets DHODH via inhibition

Developed for
COVID-19 · acute myeloid leukemia
Investigated by
Clear Creek Bio, Inc.

Trials 4 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/22 trials
Phase 1/2 NCT04425252 Aug → Dec 2020 COVID-19 Clear Creek Bio, Inc. Completed No outcome recorded
Phase 1/2 NCT03760666 Dec 2018 → Dec 2020 acute myeloid leukemia Clear Creek Bio, Inc. Terminated No outcome recorded
Phase 22 trials
Phase 2 NCT05166876 Feb → Jun 2022 COVID-19 Clear Creek Bio, Inc. Terminated No outcome recorded
Phase 2 NCT04575038 Nov 2020 → Apr 2021 COVID-19 Clear Creek Bio, Inc. Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as Brequinar ClinicalTrials.gov intervention name — accepted as the source's own label NCT04425252
3

NCT05166876

NCT04575038

NCT03760666

Known as Brequinar Sodium “Drug: Brequinar SodiumNCT05166876
Known as Brequinar sodium salt ChEMBL registry synonym — accepted as the source's own label CHEMBL38434
Known as DUP 785 ChEMBL registry synonym — accepted as the source's own label CHEMBL38434
Known as NSC-368390 ChEMBL registry synonym — accepted as the source's own label CHEMBL38434
Action Inhibit “DHODH inhibitor, 100 mg daily x 5 days” NCT04425252
Modality Small molecule CHEMBL38434
Route Oral “Brequinar and ribavirin were dosed orally” NCT03760666
Target DHODH DHODH inhibitor, 100 mg daily x 5 days” NCT04425252