Drugs / opicinumab
last change Feb 2021 re-read 2 minutes ago

opicinumab

also known as BIIB033 · Anti-LINGO · Li81

Protein / enzyme biologic targets LINGO1 via inhibition

Developed for
multiple sclerosis · optic neuritis · relapsing-remitting multiple sclerosis
Investigated by
Biogen

Trials 8 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT02833142 Jul → Nov 2016 multiple sclerosis, optic neuritis Biogen Completed No outcome recorded
Phase 1 NCT02641041 Feb → Sep 2016 multiple sclerosis Biogen Completed No outcome recorded
Phase 1 NCT01244139 Oct 2010 → Apr 2012 relapsing-remitting multiple sclerosis Biogen Completed No outcome recorded
Phase 1 NCT01052506 Jan 2010 → Oct 2011 Biogen Completed No outcome recorded
Phase 24 trials
Phase 2 NCT03222973 Nov 2017 → Feb 2021 multiple sclerosis Biogen Terminated No outcome recorded
Phase 2 NCT02657915 Mar 2016 → Jan 2017 optic neuritis Biogen Completed No outcome recorded
Phase 2 NCT01864148 Aug 2013 → Dec 2015 multiple sclerosis Biogen Completed No outcome recorded
Phase 2 NCT01721161 Dec 2012 → Oct 2014 optic neuritis Biogen Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 10 sources stand behind the page.

FieldValueCited text
Known as opicinumab “BIIB033 (opicinumab)” NCT02833142
1

NCT03222973

Known as Anti-LINGO ChEMBL registry synonym — accepted as the source's own label CHEMBL3544922
Known as BIIB033 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01244139
6

NCT02657915

NCT02641041

NCT01864148

NCT01052506

NCT02833142

NCT01721161

Known as Li81 “The anti-LINGO-1 antibody Li81 (opicinumab), which blocks LINGO-1 function and shows robust remyelinating activity in animal models” PMID 31928294 Jan 2020
Action Inhibit “blocking the function of another protein called LINGO-1” NCT01244139
Modality Protein / enzyme biologic “BIIB033 is a protein” NCT01244139
Route Intravenous “Single, escalating doses of BIIB033 (8 cohorts IV, 1 cohort SC)” NCT01052506
Route Subcutaneous “Single, escalating doses of BIIB033 (8 cohorts IV, 1 cohort SC)” NCT01052506
Target LINGO1 “blocking the function of another protein called LINGO-1” NCT01244139