Drugs / GSK1521498
last change May 2014 re-read 2 minutes ago

GSK1521498

also known as GSK1521498H

Small molecule targets OPRM1 via inhibition

Developed for
obesity disorder · alcohol dependence
Investigated by
GlaxoSmithKline · University of Cambridge

Trials 5 · a red edge is where a trial was stopped

2009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT01738867 Dec 2012 → May 2014 alcohol dependence GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT01366573 May → Sep 2011 alcohol dependence GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT00976105 Sep 2009 → Mar 2010 obesity disorder GlaxoSmithKline Completed No outcome recorded
Phase 1 NCT00976066 Jun → Dec 2009 obesity disorder GlaxoSmithKline Completed No outcome recorded
Phase 21 trial
Phase 2 NCT01195792 Sep 2010 → May 2011 obesity disorder GlaxoSmithKline Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT00857883 Comparator Nov 2008 → Aug 2009 obesity disorder GlaxoSmithKline Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as GSK1521498 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01195792
5

NCT01738867

NCT00976105

NCT00857883

NCT01366573

NCT00976066

Known as GSK1521498H ChEMBL registry synonym — accepted as the source's own label CHEMBL4297383
Action Inhibit “This may stop the natural effect of opioids” NCT00857883
1

“Mu opioid receptor antagonist” CHEMBL4297383

Modality Small molecule CHEMBL4297383
Route Oral “single oral doses of GSK1521498” NCT00976066
Target OPRM1 “Mu opioid receptor antagonist” CHEMBL4297383