Drugs / Telotristat etiprate
last change Oct 2020 re-read 2 minutes ago

Telotristat etiprate

also known as LX1606 · telotristat ethyl
Developed for
carcinoid syndrome · neuroendocrine neoplasm · ulcerative colitis
Investigated by
Lexicon Pharmaceuticals · Ipsen · Barbara Ann Karmanos Cancer Institute · National Cancer Institute (NCI)

Regulatory milestones approvals, filings & regulatory actions · 2 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved EU (EMA) Xermelo 2017-09-17 europa.eu
Approved US (FDA) XERMELO 2017-02-28 fda.gov

Trials 13 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT03442725 Feb → Apr 2018 impaired renal function disease Ipsen Completed No outcome recorded
Phase 1 NCT02683577 Feb → Jul 2016 Ipsen Completed No outcome recorded
Phase 1 NCT02195635 Jul → Oct 2014 Lexicon Pharmaceuticals Completed No outcome recorded
Phase 1 NCT02157558 Jul → Aug 2014 Lexicon Pharmaceuticals Completed No outcome recorded
Phase 1 NCT02155205 May → Aug 2014 Lexicon Pharmaceuticals Completed No outcome recorded
Phase 1 NCT02147808 May → Aug 2014 Lexicon Pharmaceuticals Completed No outcome recorded
Phase 24 trials
Phase 2 NCT03453489 Jun 2018 → Oct 2020 carcinoid syndrome, neuroendocrine neoplasm Barbara Ann Karmanos Cancer Institute Completed No outcome recorded
Phase 2 NCT01456052 Jan 2012 → Sep 2013 ulcerative colitis Lexicon Pharmaceuticals Completed No outcome recorded
Phase 2 NCT01104415 Jun 2010 → Feb 2014 carcinoid syndrome Lexicon Pharmaceuticals Completed No outcome recorded
Phase 2 NCT00853047 Mar 2009 → Jun 2014 carcinoid syndrome Lexicon Pharmaceuticals Completed No outcome recorded
Phase 33 trials
Phase 3 NCT02063659 Mar 2014 → Mar 2016 carcinoid syndrome Lexicon Pharmaceuticals Completed No outcome recorded
Phase 3 NCT02026063 Jan 2014 → Sep 2018 carcinoid syndrome Lexicon Pharmaceuticals Completed No outcome recorded
Phase 3 NCT01677910 Jan 2013 → Mar 2016 carcinoid syndrome Lexicon Pharmaceuticals Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 14 sources stand behind the page.

FieldValueCited text
Known as telotristat etiprate ClinicalTrials.gov intervention name — accepted as the source's own label NCT02683577
12

NCT01104415

NCT02147808

NCT02195635

NCT02026063

NCT00853047

NCT01677910

NCT02063659

NCT03453489

NCT01456052

NCT02157558

NCT03442725

NCT02155205

Known as LX1606 “Study of Telotristat Etiprate (LX1606) in Participants With Symptomatic Carcinoid Syndrome” NCT01104415
2

“Single Dose of Telotristat Etiprate (LX1606) 1500 mg Compared With Placebo” NCT02155205

“500 mg telotristat etiprate (LX1606) administered orally.” NCT01456052

Known as telotristat ethyl “telotristat etiprate (telotristat ethyl) treatment” NCT03453489
Action Inhibit “Telotristat etiprate, a tryptophan hydroxylase inhibitor” PMID 27041406 Mar 2016
Route Oral “Telotristat etiprate capsules; orally 3 times daily.” NCT00853047