Drugs / KPT-330

Trials 4

201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT02471911 Dec 2015 → Oct 2019 diffuse large B-cell lymphoma Weill Medical College of Cornell University Completed No outcome recorded
Phase 1 NCT02091245 Mar 2014 → Feb 2018 overdue blast phase chronic myelogenous leukemia, BCR-ABL1 positive, childhood acute lymphoblastic leukemia, mixed phenotype acute leukemia Dana-Farber Cancer Institute Active not recruiting No outcome recorded
Phase 1 NCT02078349 Feb 2014 → Mar 2020 cancer National University Hospital, Singapore Completed No outcome recorded
Phase 1 NCT01607892 Jul 2012 → Oct 2015 hematopoietic and lymphoid cell neoplasm Karyopharm Therapeutics Inc Completed No outcome recorded

Press releases naming this drug 28 releases

DateIssuerRelease
2015-11-30 Karyopharm Therapeutics Inc Karyopharm to Present Clinical Data Update for Selinexor (KPT-330) in Hematologic Malignancies karyopharm.com ↗
2015-06-01 Karyopharm Therapeutics Inc Karyopharm Presents Clinical Data for Selinexor (KPT-330) in Patients With Recurrent Glioblastoma and Advanced Sarcomas at 2015 ASCO Annual Meeting karyopharm.com ↗
2015-05-30 Karyopharm Therapeutics Inc Karyopharm Presents Clinical Data for Selinexor (KPT-330) in Patients With Heavily Pretreated Gynecological Cancers and Asian Patients With Advanced Malignancies at 2015 ASCO Annual Meeting karyopharm.com ↗
2015-05-28 Karyopharm Therapeutics Inc Karyopharm Initiates STORM Clinical Trial of Oral Selinexor (KPT-330) in Multiple Myeloma karyopharm.com ↗
2015-05-27 Karyopharm Therapeutics Inc Karyopharm to Present Clinical Data Update for Selinexor (KPT-330) in Solid Tumors karyopharm.com ↗
2015-04-13 Karyopharm Therapeutics Inc Karyopharm Granted U.S. Composition-of-Matter Patent for Selinexor (KPT-330) karyopharm.com ↗
2015-01-08 Karyopharm Therapeutics Inc Karyopharm Announces Orphan Designation Granted by FDA for Selinexor (KPT-330) in Multiple Myeloma karyopharm.com ↗
2014-12-11 Karyopharm Therapeutics Inc Karyopharm Initiates Third Registration-Directed Clinical Trial of Oral Selinexor (KPT-330) karyopharm.com ↗
2014-12-08 Karyopharm Therapeutics Inc Karyopharm Presents Positive Combination Data for Selinexor (KPT-330) in Multiple Myeloma Patients at ASH 2014 Annual Meeting karyopharm.com ↗
2014-12-08 Karyopharm Therapeutics Inc Karyopharm Presents Positive Clinical Data for Selinexor (KPT-330) in NHL Patients at ASH 2014 Annual Meeting karyopharm.com ↗
2014-12-01 Karyopharm Therapeutics Inc Karyopharm Announces Additional Orphan Designations Granted for Selinexor (KPT-330) by European Commission karyopharm.com ↗
2014-11-10 Karyopharm Therapeutics Inc Karyopharm Initiates Registration-Directed Clinical Study of Selinexor (KPT-330) in Patients With Richter's Transformation karyopharm.com ↗

Evidence & citations 4 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as KPT-330 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02471911 ↗
3

NCT02091245 ↗

NCT01607892 ↗

NCT02078349 ↗

Action Inhibit “selective inhibitor of the nuclear export protein XPO1” PMID 29203585 ↗ Dec 2017
Route Oral “for oral administration” NCT02078349 ↗
Target XPO1 “selective inhibitor of the nuclear export protein XPO1” PMID 29203585 ↗ Dec 2017