Drugs / Avanafil
last change Oct 2022 re-read 2 minutes ago

Avanafil

also known as TA-1790 · Avanafilo · Spedra · Stendra

Small molecule targets PDE5A via inhibition

Developed for
erectile dysfunction
Investigated by
VIVUS LLC · Covance · JW Pharmaceutical · Pusan National University Hospital · Sanofi

Regulatory milestones approvals, filings & regulatory actions · 6 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (3) US (FDA) STENDRA 2014-09-17 – 2022-10-18 fda.gov
Approved EU (EMA) Spedra 2013-06-21 europa.eu
Refused (EMA) EU (EMA) Spedra 2013-04-26 europa.eu
Approved US (FDA) STENDRA 2012-04-27 fda.gov

Trials 20 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 110 trials
Phase 1 NCT01095601 Apr → May 2010 VIVUS LLC Completed No outcome recorded
Phase 1 NCT01117038 Apr → May 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 1 NCT01095588 Apr → May 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 1 NCT01100021 Feb → Mar 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 1 NCT01054261 Jan → Feb 2010 VIVUS LLC Completed No outcome recorded
Phase 1 NCT01054430 Jan → Feb 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 1 NCT00914511 May → Jun 2009 VIVUS LLC Completed No outcome recorded
Phase 1 NCT00770042 Oct → Nov 2008 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 1 NCT00769041 Oct 2008 → Jan 2009 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 1 NCT01616485 Mar → May 2004 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 21 trial
Phase 2 NCT02477436 Feb → Sep 2008 erectile dysfunction Pusan National University Hospital Completed No outcome recorded
Phase 36 trials
Phase 3 NCT02503306 Jul 2015 → Mar 2016 erectile dysfunction Sanofi Completed No outcome recorded
Phase 3 NCT00895011 Apr 2009 → Apr 2011 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 3 NCT00903981 Mar → Oct 2009 erectile dysfunction JW Pharmaceutical Completed No outcome recorded
Phase 3 NCT00853606 Mar 2009 → Apr 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 3 NCT00809471 Dec 2008 → Feb 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 3 NCT00790751 Nov 2008 → Aug 2009 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 43 trials
Phase 4 NCT02033200 Jan 2014 VIVUS LLC Completed No outcome recorded
Phase 4 NCT01768676 Dec 2012 → Aug 2014 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 4 NCT01698684 Sep 2012 → Apr 2013 erectile dysfunction VIVUS LLC Completed No outcome recorded
Also used as a comparator or background therapy in 4 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT01054859 Comparator Jan 2010 erectile dysfunction VIVUS LLC Completed No outcome recorded
Phase 31 trial
Phase 3 NCT01705197 Comparator Feb 2012 → Apr 2013 erectile dysfunction JW Pharmaceutical Completed No outcome recorded
Phase 42 trials
Phase 4 NCT04374994 Comparator Sep 2018 → Apr 2019 erectile dysfunction University of Alexandria Completed No outcome recorded
Phase 4 NCT03169582 Comparator Apr 2016 → Jun 2018 erectile dysfunction Eduardo Vargas-Baquero Unknown No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 25 sources stand behind the page.

FieldValueCited text
Known as avanafil ClinicalTrials.gov intervention name — accepted as the source's own label NCT00809471
21

NCT02477436

NCT00769041

NCT01698684

NCT01100021

NCT00853606

NCT00914511

NCT00790751

NCT01054430

NCT01054261

NCT01705197

NCT00770042

NCT01095601

NCT02503306

NCT03169582

NCT00903981

NCT00895011

NCT01768676

NCT01117038

NCT01054859

NCT01095588

NCT04374994

Known as Avanafilo ChEMBL registry synonym — accepted as the source's own label CHEMBL1963681
Known as Spedra ChEMBL registry synonym — accepted as the source's own label CHEMBL1963681
Known as Stendra ClinicalTrials.gov intervention name — accepted as the source's own label NCT02033200
Known as TA-1790 “A Phase I, Single-Centre, Open-Label, Randomized, One-sequence Crossover, Three-Group Study to Evaluate the Effect of Ketoconazole, Ritonavir and Erythromicin on the Safety and...” NCT00770042
2

“AVANAFIL (TA-1790)” NCT01054430

NCT01616485

Action Inhibit “Avanafil is a potent and highly specific PDE5 inhibitor” NCT00770042
1

“Phosphodiesterase 5A inhibitor” CHEMBL1963681

Modality Small molecule CHEMBL1963681
Route Oral “30 minutes orally prior to initiation of sexual activity” NCT00790751
Target PDE5A “Phosphodiesterase 5A inhibitor” CHEMBL1963681