Drugs / Fosifloxuridine Nafalbenamide
last change May 2025 re-read 2 minutes ago

Fosifloxuridine Nafalbenamide

Other / unclassified targets TYMS via inhibition

Developed for
cancer · colorectal adenocarcinoma · colorectal carcinoma · malignant pleural mesothelioma · non-small cell lung carcinoma
Investigated by
NuCana plc · University of Oxford

Trials 4 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT02723240 Jan 2016 → Feb 2020 cancer University of Oxford Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT05714553 Mar 2023 → May 2025 cancer of unknown primary site, carcinoma of esophagus, classic Hodgkin lymphoma, colorectal cancer +11 NuCana plc Terminated No outcome recorded
Phase 1/2 NCT03428958 Oct 2018 → Mar 2024 colorectal carcinoma NuCana plc Completed No outcome recorded
Phase 21 trial
Phase 2 NCT05678257 Apr 2023 → Aug 2024 colorectal adenocarcinoma NuCana plc Terminated No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as Fosifloxuridine Nafalbenamide ClinicalTrials.gov intervention name — accepted as the source's own label NCT05714553
1

NCT05678257

Known as CPF-373 ChEMBL registry synonym — accepted as the source's own label CHEMBL2181367
Known as Fosifloxuridina nafalbenamida ChEMBL registry synonym — accepted as the source's own label CHEMBL2181367
Known as NUC-3073 ChEMBL registry synonym — accepted as the source's own label CHEMBL2181367
Known as NUC-3373 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03428958
1

NCT02723240

Action Inhibit “NUC-3373, a targeted thymidylate synthase inhibitor” PMID 38566164 Apr 2024
Modality Small molecule “NUC-3373 (a pyrimidine nucleotide analogue)” NCT02723240
Route Intravenous “administered weekly or fortnightly as an I.V. (intravenous) infusion” NCT02723240
Target TYMS “NUC-3373, a targeted thymidylate synthase inhibitor” PMID 38566164 Apr 2024