Drugs / Cinnarizine
Cinnarizine
also known as
516 MD · Aplactan · Aplexal · Artate · Carecin · Cerebolan · Cerepar · Cinaperazine · +35 more
Small molecule targets HRH1 via inhibition
Trials 3
| Phase | Registry id | Dates | Indication | Sponsor | Status | Outcome |
|---|---|---|---|---|---|---|
| Phase 41 trial | ||||||
| Phase 4 | NCT06321341 | Jan 2024 → Dec 2026 expected | dysautonomia | Valenta Pharm JSC | Recruiting | No outcome recorded |
| Phase not applicable2 trials · 1 missed | ||||||
| — | NCT05686993 | Apr → Sep 2023 | primary aldosteronism, secondary hypertension | Queen Mary University of London | Completed | Missed primary |
| — | NCT01198106 | Sep 2009 → Sep 2010 | motion sickness | Medical Corps, Israel Defense Force | Unknown | No outcome recorded |
| Comparator or background therapy1 trial | ||||||
| Phase 4 | NCT01939093 Background | Mar 2010 → Sep 2011 | methamphetamine-induced psychosis | Chulalongkorn University | Completed | No outcome recorded |
Evidence & citations 48 cited values
Every value below carries the sentence it was read from. 6 sources stand behind the page.
| Field | Value | Cited text |
|---|---|---|
| Known as | cinnarizine | “Dimenhydrinate + Cinnarizine” NCT06321341 ↗ |
| Known as | 516 MD | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Aplactan | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Aplexal | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Artate | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Carecin | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cerebolan | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cerepar | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinaperazine | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinarizina | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinarizine | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinazyn | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinnacet | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinnageron | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Cinnipirine | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Corathiem | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Denapol | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Dimitron | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Eglen | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Folcodal | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Giganten | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Glanil | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Hilactan | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Ixertol | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Katoseran | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Labyrin | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Marzine r.f. | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Midronal | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Mitronal | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Mylan travel sickness | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | NSC-758400 | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Olamin | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Processine | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | R 1575 | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | R 516 | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Sedatromin | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Sepan | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Siptazin | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Spaderizine | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Stugeron | ClinicalTrials.gov intervention name — accepted as the source's own label NCT01939093 ↗ |
| Known as | Stugeron fte | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Stunarone | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Stutgeron | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Known as | Stutgin | ChEMBL registry synonym — accepted as the source's own label CHEMBL43064 ↗ |
| Action | Inhibit | “Cav1.3 blockade by cinnarizine may achieve similar, or greater, reduction in aldosterone secretion than nonselective Cav1.2/1.3 blockade by nifedipine.” PMID 40052842 ↗ Sep 20251“Histamine H1 receptor antagonist” CHEMBL43064 ↗ |
| Modality | Small molecule | — CHEMBL43064 ↗ |
| Route | Oral | “oral cinnarizine” NCT01198106 ↗ |
| Target | HRH1 | “Histamine H1 receptor antagonist” CHEMBL43064 ↗ |