Drugs / CARBETAPENTANE
CARBETAPENTANE
also known as
CARBETAPENTANE CITRATE · Loucarbate · NSC-757833 · Pentoxiverina · pentoxyverine · pentoxyverine citrate · Pentoxyverine hydrogen citrate · Sedotussin · +1 more
Small molecule targets SIGMAR1 via activation
Trials 1
| Phase | Registry id | Dates | Indication | Sponsor | Status | Outcome |
|---|---|---|---|---|---|---|
| Phase 1 | NCT02183649 | Nov → Dec 2009 | — | Boehringer Ingelheim | Completed | No outcome recorded |
Evidence & citations 14 cited values
Every value below carries the sentence it was read from. 2 sources stand behind the page.
| Field | Value | Cited text |
|---|---|---|
| Known as | CARBETAPENTANE | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | CARBETAPENTANE CITRATE | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | Loucarbate | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | NSC-757833 | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | Pentoxiverina | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | pentoxyverine | ClinicalTrials.gov intervention name — accepted as the source's own label NCT02183649 ↗ |
| Known as | pentoxyverine citrate | “192 mg Pentoxyverine Citrate (Corresponding to 121.5 mg Pentoxyverine Base)” NCT02183649 ↗ |
| Known as | Pentoxyverine hydrogen citrate | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | Sedotussin | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Known as | Toclase | ChEMBL registry synonym — accepted as the source's own label CHEMBL73234 ↗ |
| Action | Activate | “Sigma opioid receptor agonist” CHEMBL73234 ↗ |
| Modality | Small molecule | — CHEMBL73234 ↗ |
| Route | Oral | “After a Single Oral Dose” NCT02183649 ↗ |
| Target | SIGMAR1 | “Sigma opioid receptor agonist” CHEMBL73234 ↗ |